SCHEMBL8564247

SCHEMBL8564247

CCCCOC(=O)n1cc(S(=O)(=O)Cl)c2ccc(-c3ccc(F)cc3)cc21

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ASAH1 Q13510 3/20 0.39
SERPINE1 P05121 1/20 0.35
GSK3B P49841 1/20 0.34
BCHE P06276 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34
GRIN2B Q13224 1/20 0.34
CHRNA7 P36544 1/20 0.34
RARA P10276 1/20 0.33
RARB P10826 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7845141 0.82 HDAC2 (0.39) SERPINE1GRIN2B
SCHEMBL9054223 0.74 HTT (0.42)
SCHEMBL28743917 0.70 BCHE (0.45) BCHEALDH1A1KMT2ATP53MAPT
SCHEMBL8564251 0.69 GPR17 (0.42) GSK3BALDH1A1KMT2A
SCHEMBL30622564 0.66 NPC1 (0.39) BCHEALDH1A1KMT2A
SCHEMBL30182164 0.65 KMT2A (0.36) ASAH1BCHEALDH1A1KMT2ATP53
SCHEMBL1553715 0.65 SLC22A12 (0.47) RARBTP53
SCHEMBL124286 0.65 HDAC2 (0.41) SERPINE1GRIN2B
SCHEMBL8570658 0.63 TSHR (0.47) GSK3BALDH1A1KMT2ATP53
SCHEMBL8083502 0.62 BCHE (0.49) BCHEALDH1A1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821685-A1 INDOLE-3-CARBONYL AND INDOLE-3-SULFONYL DERIVATIVES AS PLATELET ACTIVATING FACTOR ANTAGONISTS ABBOTT LABORATORIES (US) 1998-02-04 EP disclosed