SCHEMBL8564261

SCHEMBL8564261

COc1ccc(N)c(-n2cccc2)n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.34
GAA P10253 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.34
SIRT1 Q96EB6 1/20 0.34
NNMT P40261 1/20 0.34
JAK2 O60674 1/20 0.34
ALDH1A1 P00352 3/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
MTNR1A P48039 2/20 0.32
MTNR1B P49286 2/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32
USP7 Q93009 1/20 0.32
TDP1 Q9NUW8 2/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4119372 0.76 CYP1A2 (0.36) SIRT2SIRT1NNMTPDE10ACYP1A2
SCHEMBL2266765 0.74 CASP3 (0.44) KDM4EALDH1A1RAB9AMAPTHPGD
SCHEMBL2267089 0.72 HTR2A (0.43) SIRT2SIRT1NNMTHTR2AHTR2C
SCHEMBL5752945 0.72 ALDH1A1 (0.45) KDM4EGAAALDH1A1RAB9AMAPT
Hydrochloric Acid SCHEMBL6261576 0.72 CASP3 (0.43) KDM4EALDH1A1MAPTHPGDHSD17B10
SCHEMBL8569551 0.72 TXNRD1 (0.50) JAK2RAB9AMAPT
SCHEMBL8570449 0.72 POLB (0.41) KDM4EGAASIRT2ALDH1A1NPC1
SCHEMBL5751466 0.71 HRH4 (0.51) KDM4EGAAALDH1A1MAPTHPGD
SCHEMBL2270412 0.70 GAA (0.47) KDM4EGAAALDH1A1MAPTHPGD
SCHEMBL2267531 0.70 CHRNB2 (0.47) KDM4EALDH1A1MAPTHPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623620-B1 5-HT3 Pyrrolopyrazine derivatives ADIR (FR) 1998-09-09 EP disclosed
US-5599812-A ANTISEROTONINE AGENTS ADIR ET COMPAGNIE (FR) 1997-02-04 US disclosed
EP-0623620-A1 5-HT3 Pyrrolopyrazine derivatives ADIR ET COMPAGNIE (FR) 1994-11-09 EP disclosed