SCHEMBL8564795

SCHEMBL8564795

COc1ccc2[nH]c(-c3cccc4ccccc34)nc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.50
RAB9A P51151 6/20 0.50
KDM4E B2RXH2 5/20 0.50
SMN1; SMN2 Q16637 5/20 0.50
ALDH1A1 P00352 4/20 0.50
HPGD P15428 4/20 0.50
HSD17B10 Q99714 2/20 0.50
TP53 P04637 2/20 0.50
TSHR P16473 1/20 0.50
NFKB1 P19838 1/20 0.50
NFKB2 Q00653 1/20 0.50
RELA Q04206 1/20 0.50
PKM P14618 2/20 0.49
GUSB P08236 1/20 0.48
AMY1A P0DUB6 4/20 0.48
MAPT P10636 4/20 0.47
GLA P06280 1/20 0.47
GAA P10253 1/20 0.47
RECQL P46063 1/20 0.47
MEN1 O00255 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4496832 0.89 NPC1 (0.57) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL4496843 0.83 NPC1 (0.68) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL22955586 0.83 RUNX1 (0.49) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL14876858 0.83 ABCG2 (0.52) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL19205885 0.82 GUSB (0.55) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL22955874 0.82 ALDH1A1 (0.52) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL1170729 0.81 ALDH1A1 (0.57) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL14876859 0.81 GUSB (0.63) NPC1RAB9AKDM4EHSD17B10GUSB
SCHEMBL27824953 0.80 HPGD (0.47) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL8108604 0.80 NPC1 (0.69) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021022061-A1 ARYL HYDROCARBON RECEPTOR ACTIVATORS OREGON STATE UNIVERSITY (US) 2021-02-04 WO disclosed
EP-0821675-A1 NOVEL HYDROXAMIC ACID AND AMINO-CARBOXYLATE COMPOUNDS AS METALLOPROTEASE AND TNF INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-02-04 EP disclosed
WO-1996033176-A1 NOVEL HYDROXAMIC ACID AND AMINO-CARBOXYLATE COMPOUNDS AS METALLOPROTEASE AND TNF INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-10-24 WO disclosed