SCHEMBL8564818

SCHEMBL8564818

CC1(C)NCCc2cc(N3C(=O)NCC3c3ccc(CCC(=O)O)cc3)ccc21

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.39
CYP26B1 Q9NR63 4/20 0.39
CYP26A1 O43174 3/20 0.39
CYP3A4 P08684 1/20 0.35
QPCT Q16769 13/20 0.35
QPCTL Q9NXS2 1/20 0.35
PPARD Q03181 1/20 0.32
PPARA Q07869 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562406 0.85 HTR6 (0.39) QPCTQPCTLPPARDPPARA
SCHEMBL8564812 0.84 ESR1 (0.31) ESR1QPCT
SCHEMBL8557055 0.83 ITGB3 (0.38) QPCTQPCTLPPARDPPARA
SCHEMBL8559860 0.82 PARP1 (0.39) ESR1CYP26B1CYP26A1QPCTQPCTL
Hydrochloric Acid SCHEMBL8563477 0.81 PARP1 (0.38) ESR1CYP26B1CYP26A1QPCTQPCTL
Hydrochloric Acid SCHEMBL8559595 0.80 QPCT (0.37) ESR1QPCTQPCTL
SCHEMBL8559323 0.80 PARP1 (0.37) ESR1QPCTQPCTL
SCHEMBL8560495 0.80 HTR6 (0.43) ESR1QPCTQPCTLPPARDPPARA
SCHEMBL8562965 0.79 ESR1 (0.44) ESR1CYP26B1CYP26A1CYP3A4PPARD
Hydrochloric Acid SCHEMBL8565143 0.79 QPCT (0.37) ESR1CYP26B1CYP26A1QPCTQPCTL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed