SCHEMBL8564870

SCHEMBL8564870

Clc1ccc2nc(Cl)c3cccn3c2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 3/20 0.40
HTR3E A5X5Y0 8/20 0.38
HTR3B O95264 8/20 0.38
HTR3A P46098 8/20 0.38
HTR3D Q70Z44 8/20 0.38
HTR3C Q8WXA8 8/20 0.38
RPS6KA5 O75582 1/20 0.36
RPS6KA4 O75676 1/20 0.36
HTR1A P08908 6/20 0.35
PTPN2 P17706 1/20 0.35
KDM4E B2RXH2 4/20 0.35
ALDH1A1 P00352 4/20 0.35
HPGD P15428 4/20 0.35
GLA P06280 3/20 0.35
GAA P10253 3/20 0.35
POLB P06746 2/20 0.35
HSD17B10 Q99714 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HTR2C P28335 3/20 0.34
MEN1 O00255 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8563939 0.80 HTR3E (0.55) PTPN1HTR3EHTR3BHTR3AHTR3D
SCHEMBL8570625 0.78 HTR3E (0.55) PTPN1HTR3EHTR3BHTR3AHTR3D
SCHEMBL4040875 0.75 BTK (0.39) RPS6KA5RPS6KA4HRH4
SCHEMBL8569855 0.74 PTPN1 (0.61) PTPN1HTR3EHTR3BHTR3AHTR3D
SCHEMBL8563514 0.73 HTR3E (0.65) PTPN1HTR3EHTR3BHTR3AHTR3D
SCHEMBL2460828 0.72 PTPN1 (0.71) PTPN1HTR3EHTR3BHTR3AHTR3D
SCHEMBL8567409 0.70 HTR3E (0.38) PTPN1HTR3EHTR3BHTR3AHTR3D
SCHEMBL7401133 0.69 PTPN1 (0.54) PTPN1HTR3EHTR3BHTR3AHTR3D
SCHEMBL14828916 0.69 HRH4 (0.54) ALDH1A1POLBMEN1KMT2AHRH4
SCHEMBL8565857 0.68 PARP1 (0.53) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623620-B1 5-HT3 Pyrrolopyrazine derivatives ADIR (FR) 1998-09-09 EP disclosed
US-5599812-A ANTISEROTONINE AGENTS ADIR ET COMPAGNIE (FR) 1997-02-04 US disclosed
EP-0623620-A1 5-HT3 Pyrrolopyrazine derivatives ADIR ET COMPAGNIE (FR) 1994-11-09 EP disclosed