SCHEMBL8570625

SCHEMBL8570625

Clc1nc2cccnc2n2cccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 9/20 0.55
HTR3B O95264 9/20 0.55
HTR3A P46098 9/20 0.55
HTR3D Q70Z44 9/20 0.55
HTR3C Q8WXA8 9/20 0.55
HTR1A P08908 7/20 0.55
HTR2C P28335 6/20 0.55
RPS6KA5 O75582 3/20 0.41
RPS6KA4 O75676 1/20 0.41
PDE2A O00408 1/20 0.39
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
PTPN2 P17706 1/20 0.38
PTPN1 P18031 1/20 0.38
RAD51 Q06609 1/20 0.37
CYP1A2 P05177 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8567409 0.79 HTR3E (0.38) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL8564870 0.78 PTPN1 (0.40) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL4038518 0.78 LCK (0.41) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL8569855 0.77 PTPN1 (0.61) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL30578099 0.75 MAPK8 (0.54) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL120846 0.75 MAPK8 (0.54) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL8563997 0.74 HTR3E (0.78) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL8561755 0.73 HTR3E (0.80) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL8570035 0.73 HTR3E (0.54) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL21208491 0.72 TYMS (0.50) PDE2AKDM4EALDH1A1GLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623620-B1 5-HT3 Pyrrolopyrazine derivatives ADIR (FR) 1998-09-09 EP disclosed
US-5599812-A ANTISEROTONINE AGENTS ADIR ET COMPAGNIE (FR) 1997-02-04 US disclosed
EP-0623620-A1 5-HT3 Pyrrolopyrazine derivatives ADIR ET COMPAGNIE (FR) 1994-11-09 EP disclosed