SCHEMBL8564897

SCHEMBL8564897

CNc1nc(Cl)c(Sc2cccc(Cl)c2)c(Cl)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.49
DRD2 P14416 1/20 0.49
DRD4 P21917 1/20 0.49
TYMS P04818 3/20 0.44
HPGD P15428 4/20 0.41
KDM4E B2RXH2 3/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
ADORA1 P30542 1/20 0.41
XBP1 P17861 1/20 0.41
DHFR P00374 2/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 3/20 0.40
POLB P06746 1/20 0.39
MAPT P10636 2/20 0.39
SLC6A2 P23975 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8564591 0.83 HTR1A (0.64) HTR1ADRD2DRD4TYMSHPGD
SCHEMBL8563375 0.82 HTR1A (0.79) HTR1ADRD2DRD4
SCHEMBL8571069 0.82 KDM4E (0.45) TYMSHPGDKDM4ELMNACYP1A2
SCHEMBL8570657 0.80 HTR1A (0.50) HTR1ADRD2DRD4TYMSHPGD
SCHEMBL29543630 0.71 POLB (0.56) HPGDKDM4ELMNACYP1A2CYP3A4
SCHEMBL30688805 0.71 POLB (0.56) HPGDKDM4ELMNACYP1A2CYP3A4
SCHEMBL2282611 0.71 POLB (0.56) HPGDKDM4ELMNACYP1A2CYP3A4
SCHEMBL10596007 0.69 POLB (0.55) HPGDKDM4ELMNACYP1A2CYP3A4
SCHEMBL27999929 0.68 SLC6A2 (0.54) HPGDKDM4ELMNACYP1A2CYP3A4
SCHEMBL10708413 0.67 POLB (0.62) HPGDKDM4ELMNACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0826674-A1 NOVEL PYRIMIDINE DERIVATIVES EFFICACIOUS AS PSYCHOTROPIC DRUG AND PROCESS FOR THE PRODUCTION THEREOF SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1998-03-04 EP disclosed