SCHEMBL8565077

SCHEMBL8565077

COc1ccc(OCC(N)=O)c(N)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.56
KMT2A Q03164 3/20 0.56
MEN1 O00255 2/20 0.56
MAPT P10636 2/20 0.56
THRB P10828 2/20 0.56
SNCA P37840 1/20 0.48
KDM4E B2RXH2 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
GAA P10253 1/20 0.46
RECQL P46063 1/20 0.46
BLM P54132 1/20 0.46
MCL1 Q07820 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
LMNA P02545 2/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8569529 0.87 ALDH1A1 (0.56) ALDH1A1KMT2AMEN1MAPTTHRB
SCHEMBL4612728 0.87 PTGDR2 (0.57) ALDH1A1KMT2AMEN1MAPTTHRB
SCHEMBL656717 0.87 MEN1 (0.56) ALDH1A1KMT2AMEN1MAPTTHRB
SCHEMBL15330191 0.80 KDM4E (0.67) ALDH1A1KMT2AMEN1MAPTSNCA
SCHEMBL15933189 0.80 KDM4E (0.51) ALDH1A1KMT2AMEN1MAPTSNCA
SCHEMBL6536100 0.78 LMNA (0.54) ALDH1A1KMT2AMEN1MAPTTHRB
SCHEMBL8562385 0.78 USP2 (0.58) ALDH1A1MAPTKDM4ESMN1; SMN2GAA
SCHEMBL28950410 0.78 ALDH1A1 (0.61) ALDH1A1KMT2AMEN1MAPTTHRB
SCHEMBL11212890 0.78 KMT2A (0.57) ALDH1A1KMT2AMEN1MAPTSNCA
SCHEMBL8569607 0.78 RAB9A (0.56) ALDH1A1KMT2AMEN1MAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719141-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1998-02-17 US disclosed
EP-0702004-A2 2,9-diamino- and 2-amino-8-carbamoyl-4-hydroxy-alkanoic acid amid derivatives CIBA-GEIGY AG (CH) 1996-03-20 EP disclosed