SCHEMBL8565096

SCHEMBL8565096

O=C1Nc2ccccc2C(c2ccccc2)N1C1CCN(Cc2ccncc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 2/20 0.48
TRPV6 Q9H1D0 1/20 0.48
SIGMAR1 Q99720 1/20 0.47
OPRL1 P41146 2/20 0.45
ACHE P22303 1/20 0.43
CHRM3 P20309 5/20 0.43
CHRM2 P08172 4/20 0.43
KDM1A O60341 1/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6168606 0.92 OPRL1 (0.52) CCR5OPRL1ACHECHRM3CHRM2
SCHEMBL29445321 0.92 OPRL1 (0.52) CCR5OPRL1ACHECHRM3CHRM2
SCHEMBL8570739 0.90 CHRM2 (0.54) CCR5TRPV6SIGMAR1OPRL1ACHE
SCHEMBL8565038 0.88 CHRM3 (0.47) CCR5TRPV6SIGMAR1OPRL1ACHE
SCHEMBL8569508 0.88 MEN1 (0.53) CCR5SIGMAR1OPRL1ACHECHRM3
SCHEMBL6168165 0.86 CHRM3 (0.49) SIGMAR1OPRL1ACHECHRM3CHRM2
SCHEMBL8570369 0.85 CHRM3 (0.50) OPRL1ACHECHRM3CHRM2
SCHEMBL8570694 0.85 PARP1 (0.49) TRPV6SIGMAR1OPRL1CHRM3CHRM2
SCHEMBL6167277 0.85 CHRM3 (0.53) SIGMAR1OPRL1ACHECHRM3CHRM2
SCHEMBL8563897 0.84 OPRL1 (0.43) CCR5OPRL1ACHECHRM3CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626373-B1 Quinazolinone derivatives SUMITOMO PHARMA (JP) 1998-12-23 EP disclosed
US-5556860-A ANTIISCHEMIC AGENTS, BRAIN DISORDERS AND BLOOD METAL CONCENTRATIONS AND KIDNEY DISEASE SUMITOMO PHARMACEUTICALS CO., LTD. (JP) 1996-09-17 US disclosed
EP-0626373-A1 Quinazolinone derivatives SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1994-11-30 EP disclosed