SCHEMBL8565197

SCHEMBL8565197

CC(=O)N1CCCNCC1CCC(O)(c1ccccc1)c1cccc(O)c1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 10/20 0.42
CHRM3 P20309 4/20 0.37
CHRM2 P08172 3/20 0.37
CYP2D6 P10635 2/20 0.35
MAPK1 P28482 1/20 0.35
CHRM1 P11229 2/20 0.34
LMNA P02545 1/20 0.34
HTR1A P08908 1/20 0.34
OPRM1 P35372 1/20 0.34
KCNH2 Q12809 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
KIF11 P52732 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6765644 0.71 CHRM2 (0.60) CCR2CHRM3CHRM2CYP2D6MAPK1
SCHEMBL18623050 0.70 CHRM3 (0.54) CCR2CHRM3CHRM2CYP2D6CHRM1
SCHEMBL6765350 0.69 CCR2 (0.63) CCR2CHRM2CYP2D6MAPK1CHRM1
SCHEMBL5061378 0.64 KMT2A (0.56) CHRM3CHRM2CYP2D6MAPK1CHRM1
SCHEMBL25698254 0.63 HCRTR1 (0.47)
SCHEMBL7808926 0.63 KIF11 (0.47) CCR2LMNAKIF11
SCHEMBL3576211 0.62 CA1 (0.54)
SCHEMBL2086686 0.62 CA1 (0.54)
SCHEMBL18632724 0.62 ACHE (0.44) CCR2CHRM3CHRM2CYP2D6CHRM1
SCHEMBL27803558 0.61 CA1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997044329-A9 DIARYLALKYL CYCLIC DIAMINE DERIVATIVES AS CHEMOKINE RECEPTOR ANTAGONISTS 1998-03-12 WO disclosed