SCHEMBL8565477

SCHEMBL8565477

C=C[C@H](C[C@H](O)[C@H](CC(C)(C)CCO[Si](C(C)C)(C(C)C)C(C)C)NC(=O)OC(C)(C)C)C(C)C

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA7 P43166 2/20 0.38
CYP2D6 P10635 1/20 0.35
PSEN1 P49768 2/20 0.33
PSEN2 P49810 2/20 0.33
APH1B Q8WW43 2/20 0.33
NCSTN Q92542 2/20 0.33
APH1A Q96BI3 2/20 0.33
PSENEN Q9NZ42 2/20 0.33
KLK5 Q9Y337 1/20 0.32
CA4 P22748 1/20 0.31
CA9 Q16790 1/20 0.31
CTSK P43235 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8565474 1.00 CA1 (0.38) CA1CA2CA7CYP2D6PSEN1
SCHEMBL8561163 0.84 CA1 (0.36) CA1CA2CA7CYP2D6PSEN1
SCHEMBL8561160 0.84 CA1 (0.36) CA1CA2CA7CYP2D6PSEN1
SCHEMBL8569503 0.80 CYP2D6 (0.39) CA1CA2CA7CYP2D6KLK5
SCHEMBL8569499 0.80 CYP2D6 (0.39) CA1CA2CA7CYP2D6KLK5
SCHEMBL8564217 0.79 PPARA (0.45) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8564212 0.79 PPARA (0.45) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8626962 0.77 REN (0.42)
SCHEMBL8562274 0.74 CTSK (0.48) CA1CA2CA7CYP2D6CTSK
SCHEMBL8562271 0.74 CTSK (0.48) CA1CA2CA7CYP2D6CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719141-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1998-02-17 US disclosed