SCHEMBL8558614

SCHEMBL8558614

CC(C)OC(=O)CCc1ccc(N2CCN(c3ccc4c(c3)CCNCC4)C2=O)cc1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 8/20 0.38
FAAH O00519 2/20 0.36
NOTUM Q6P988 1/20 0.35
S1PR1 P21453 1/20 0.35
MLNR O43193 3/20 0.35
CYP2D6 P10635 1/20 0.35
DRD2 P14416 2/20 0.34
DRD3 P35462 2/20 0.34
KCNH2 Q12809 1/20 0.34
HRH3 Q9Y5N1 1/20 0.33
HTR2C P28335 2/20 0.33
HTR2A P28223 1/20 0.33
MCHR1 Q99705 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8568700 0.99 HTR6 (0.38) HTR6FAAHNOTUMS1PR1MLNR
SCHEMBL8565812 0.90 NOTUM (0.39) HTR6FAAHNOTUMS1PR1CYP2D6
Hydrochloric Acid SCHEMBL8559741 0.89 NOTUM (0.38) HTR6FAAHNOTUMS1PR1CYP2D6
SCHEMBL8559578 0.89 HTR6 (0.42) HTR6S1PR1MLNRDRD2DRD3
Hydrochloric Acid SCHEMBL8566255 0.88 HTR6 (0.41) HTR6S1PR1MLNRDRD2DRD3
SCHEMBL8562408 0.84 S1PR1 (0.44) HTR6S1PR1MLNR
SCHEMBL8563370 0.83 ASIC3 (0.40) HTR6S1PR1HRH3
SCHEMBL8564139 0.83 PTGER1 (0.35) HTR6FAAHS1PR1MLNR
Hydrochloric Acid SCHEMBL8567567 0.82 PTGER1 (0.36) HTR6FAAHS1PR1MLNR
Hydrochloric Acid SCHEMBL8563262 0.81 HTR6 (0.38) HTR6MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP claimed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP claimed
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP disclosed
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP disclosed