SCHEMBL8565911

SCHEMBL8565911

CCOc1cc2c(Nc3ccc(OCC(O)CO)cc3)ccnc2nc1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 15/20 0.39
CDK2 P24941 14/20 0.39
CDK1 P06493 1/20 0.38
CCNE1 P24864 1/20 0.38
EHMT2 Q96KQ7 1/20 0.37
PDGFRA P16234 2/20 0.36
DAPK3 O43293 1/20 0.36
JAK2 O60674 1/20 0.36
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
PAK4 O96013 1/20 0.36
ABL1 P00519 1/20 0.36
LCK P06239 1/20 0.36
FYN P06241 1/20 0.36
CSF1R P07333 1/20 0.36
IGF1R P08069 1/20 0.36
PDGFRB P09619 1/20 0.36
FGFR1 P11362 1/20 0.36
PRKACA P17612 1/20 0.36
LTK P29376 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8558006 0.99 CDK4 (0.38) CDK4CDK2CDK1CCNE1EHMT2
SCHEMBL8559967 0.83 PDGFRA (0.48) EHMT2PDGFRAABL1LCKACVR1
Water SCHEMBL8328226 0.82 PDGFRA (0.47) EHMT2PDGFRALCKSLC2A1
Hydrochloric Acid SCHEMBL8566059 0.82 HTT (0.50) EHMT2PDGFRALCKSLC2A1
SCHEMBL8567323 0.82 MAPKAPK2 (0.46) CDK4CDK2EHMT2PDGFRALCK
SCHEMBL8560347 0.81 ERBB2 (0.52) EHMT2PDGFRBKDRSLC2A1
Hydrochloric Acid SCHEMBL8566240 0.80 ERBB2 (0.51) EHMT2PDGFRBKDRSLC2A1
SCHEMBL8568868 0.79 HRH3 (0.49) CDK4EHMT2ABL1LCKKDR
SCHEMBL8561756 0.79 MAPT (0.51) SLC2A1
Hydrochloric Acid SCHEMBL8565861 0.78 MAPT (0.51) SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618916-B1 ANTI-RHEUMATIC NAPHTHYRIDINE DERIVATIVES KNOLL AG (DE) 1998-09-23 EP disclosed
US-5464781-A TREATING RHEUMATIC DISEASES THE BOOTS COMPANY PLC (GB) 1995-11-07 US disclosed
WO-1993013097-A1 ANTI-RHEUMATIC NAPHTHYRIDINE DERIVATIVES THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed