SCHEMBL8566129

SCHEMBL8566129

COC(=O)[C@H]1CNc2ccccc2C1=O

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
EPHX2 P34913 1/20 0.37
IDH1 O75874 1/20 0.37
MAPT P10636 1/20 0.37
ITGA4 P13612 1/20 0.37
KCNH2 Q12809 1/20 0.37
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
IDO1 P14902 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8566128 1.00 BACE1 (0.39) BACE1ALDH1A1KDM4EPOLBHPGD
SCHEMBL8566125 1.00 BACE1 (0.39) BACE1ALDH1A1KDM4EPOLBHPGD
SCHEMBL17348461 0.84 KDM4E (0.50) ALDH1A1KDM4EHPGDHSD17B10MAPT
SCHEMBL16772300 0.83 MTNR1A (0.38) ALDH1A1KDM4EHPGDHSD17B10EPHX2
SCHEMBL3830913 0.81 ALDH1A1 (0.45) ALDH1A1KDM4EMAPTKCNH2LMNA
SCHEMBL6629846 0.80 KCNH2 (0.50) BACE1ALDH1A1EPHX2MAPTKCNH2
Hydrochloric Acid SCHEMBL9046996 0.80 ALDH1A1 (0.44) ALDH1A1KDM4EMAPTKCNH2LMNA
SCHEMBL444604 0.80 LMNA (0.38) ALDH1A1KDM4EHSD17B10MAPTKCNH2
Hydrochloric Acid SCHEMBL2258244 0.78 KCNH2 (0.49) BACE1ALDH1A1EPHX2MAPTKCNH2
Hydrazine SCHEMBL27885781 0.78 ALDH1A1 (0.43) ALDH1A1KDM4EMAPTLMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719141-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1998-02-17 US disclosed
EP-0702004-A2 2,9-diamino- and 2-amino-8-carbamoyl-4-hydroxy-alkanoic acid amid derivatives CIBA-GEIGY AG (CH) 1996-03-20 EP disclosed