SCHEMBL8566372

SCHEMBL8566372

Cc1ccnc(-n2cccc2)c1[N+](=O)[O-]

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
TDP1 Q9NUW8 2/20 0.47
TSHR P16473 3/20 0.42
MAPT P10636 2/20 0.36
ATM Q13315 1/20 0.36
HPGD P15428 1/20 0.36
POLB P06746 1/20 0.36
LMNA P02545 1/20 0.36
PKM P14618 1/20 0.36
KMT2A Q03164 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
MEN1 O00255 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL843559 0.73 ALDH1A1 (0.54) ALDH1A1TDP1TSHRMAPTHPGD
SCHEMBL30197316 0.73 ALDH1A1 (0.54) ALDH1A1TDP1TSHRMAPTHPGD
SCHEMBL6276159 0.73 ADRB1 (0.48) MAPTCYP1A2CYP2C9CYP2C19
Ammonia Solution, Strong SCHEMBL27851817 0.72 ALDH1A1 (0.52) ALDH1A1TDP1TSHRMAPTHPGD
SCHEMBL28301520 0.71 CYP1A2 (0.61) ALDH1A1TDP1MAPTPOLBLMNA
SCHEMBL4053942 0.70 ALDH1A1 (0.50) ALDH1A1TDP1TSHRMAPTHPGD
SCHEMBL8563735 0.70 NOS2 (0.50) ALDH1A1MAPTHPGDLMNAKMT2A
SCHEMBL801243 0.70 ALDH1A1 (0.50) ALDH1A1TDP1TSHRMAPTHPGD
SCHEMBL31020500 0.70 ALDH1A1 (0.50) ALDH1A1TDP1TSHRMAPTHPGD
SCHEMBL29674727 0.70 NOS2 (0.50) ALDH1A1TDP1TSHRMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623620-B1 5-HT3 Pyrrolopyrazine derivatives ADIR (FR) 1998-09-09 EP disclosed
US-5599812-A ANTISEROTONINE AGENTS ADIR ET COMPAGNIE (FR) 1997-02-04 US disclosed
EP-0623620-A1 5-HT3 Pyrrolopyrazine derivatives ADIR ET COMPAGNIE (FR) 1994-11-09 EP disclosed