SCHEMBL8567153

SCHEMBL8567153

CCOC(=O)c1nc(C)c(Sc2ccccc2)n1COCc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1D P48730 1/20 0.42
MAPT P10636 4/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
ALDH1A1 P00352 6/20 0.40
POLB P06746 3/20 0.40
TDP1 Q9NUW8 2/20 0.40
MEN1 O00255 1/20 0.39
HSP90AA1 P07900 1/20 0.39
KMT2A Q03164 1/20 0.39
TSHR P16473 4/20 0.38
ATM Q13315 1/20 0.38
MAPK1 P28482 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38
TUBA1B P68363 1/20 0.38
TUBA4A P68366 1/20 0.38
TUBB4B P68371 1/20 0.38
TUBB3 Q13509 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nitric Acid SCHEMBL8566793 0.94 ALDH1A1 (0.39) CSNK1DMAPTSMN1; SMN2ALDH1A1POLB
SCHEMBL8567357 0.87 ALDH1A1 (0.38) CSNK1DMAPTSMN1; SMN2ALDH1A1POLB
SCHEMBL8568227 0.80 ALDH1A1 (0.39) CSNK1DMAPTSMN1; SMN2ALDH1A1POLB
SCHEMBL8562572 0.79 ALDH1A1 (0.38) CSNK1DSMN1; SMN2ALDH1A1POLBMEN1
SCHEMBL8567515 0.79 VCP (0.41) SMN1; SMN2ALDH1A1POLBTSHRL3MBTL1
SCHEMBL9050612 0.79 ALDH1A1 (0.40) SMN1; SMN2ALDH1A1POLBMEN1KMT2A
Hydrochloric Acid SCHEMBL8563542 0.76 ALDH1A1 (0.39) MAPTSMN1; SMN2ALDH1A1POLBMEN1
SCHEMBL8560120 0.69 ALDH1A1 (0.38) MAPTSMN1; SMN2ALDH1A1TDP1KMT2A
SCHEMBL10004802 0.69 KMT2A (0.44) CSNK1DMAPTSMN1; SMN2ALDH1A1MEN1
SCHEMBL9051616 0.68 ALDH1A1 (0.40) ALDH1A1TSHRMAPK1L3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0552060-B1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO (JP) 1998-11-18 EP disclosed
EP-0700911-A1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO., LTD. (JP) 1996-03-13 EP disclosed
US-5472965-A Useful for treatment of retrovirus infections; less toxic SHIONOGI & CO., LTD. (JP) 1995-12-05 US disclosed
US-5326780-A Acquired immunodeficiency syndrome SHIONOGI & CO., LTD. (JP) 1994-07-05 US disclosed
EP-0552060-A1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO., LTD. (JP) 1993-07-21 EP disclosed