SCHEMBL9051616

SCHEMBL9051616

Brc1nc(Br)n(COCc2ccccc2)c1Sc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
TSHR P16473 1/20 0.37
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
VCP P55072 2/20 0.34
USP2 O75604 1/20 0.33
MAPK1 P28482 1/20 0.33
ADORA2A P29274 2/20 0.31
ADORA1 P30542 1/20 0.31
LMNA P02545 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562834 0.87 ALDH1A1 (0.44) ALDH1A1TSHRCYP2C9CYP2C19VCP
SCHEMBL8567515 0.75 VCP (0.41) ALDH1A1TSHRCYP2C9CYP2C19VCP
SCHEMBL9050612 0.75 ALDH1A1 (0.40) ALDH1A1TSHRCYP2C9CYP2C19VCP
SCHEMBL8568227 0.74 ALDH1A1 (0.39) ALDH1A1TSHRCYP2C9CYP2C19VCP
SCHEMBL8562572 0.73 ALDH1A1 (0.38) ALDH1A1TSHRCYP2C9CYP2C19VCP
SCHEMBL8560120 0.72 ALDH1A1 (0.38) ALDH1A1TSHRCYP2C9CYP2C19VCP
Hydrochloric Acid SCHEMBL8563542 0.70 ALDH1A1 (0.39) ALDH1A1TSHRCYP2C9CYP2C19VCP
SCHEMBL8567357 0.69 ALDH1A1 (0.38) ALDH1A1TSHRCYP2C9CYP2C19L3MBTL1
SCHEMBL8567153 0.68 CSNK1D (0.42) ALDH1A1TSHRMAPK1LMNAL3MBTL1
SCHEMBL8536161 0.68 ALDH1A1 (0.43) ALDH1A1TSHRVCPUSP2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700911-A1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO., LTD. (JP) 1996-03-13 EP disclosed
US-5472965-A Useful for treatment of retrovirus infections; less toxic SHIONOGI & CO., LTD. (JP) 1995-12-05 US disclosed
US-5326780-A Acquired immunodeficiency syndrome SHIONOGI & CO., LTD. (JP) 1994-07-05 US disclosed
EP-0552060-A1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO., LTD. (JP) 1993-07-21 EP disclosed