SCHEMBL8567357

SCHEMBL8567357

Cc1nc(C(N)=O)n(COCc2ccccc2)c1Sc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP2C9 P11712 3/20 0.35
CYP2C19 P33261 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 1/20 0.35
POLB P06746 1/20 0.35
CSNK1D P48730 1/20 0.35
TSHR P16473 1/20 0.34
RAB9A P51151 1/20 0.34
PARP1 P09874 1/20 0.34
CXCL12 P48061 1/20 0.33
PARP10 Q53GL7 1/20 0.33
TOP2A P11388 1/20 0.33
TOP2B Q02880 1/20 0.33
MAPT P10636 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
NCOA1 Q15788 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8567153 0.87 CSNK1D (0.42) ALDH1A1MEN1KMT2ASMN1; SMN2POLB
Nitric Acid SCHEMBL8566793 0.81 ALDH1A1 (0.39) ALDH1A1MEN1KMT2ASMN1; SMN2POLB
SCHEMBL8562572 0.81 ALDH1A1 (0.38) ALDH1A1MEN1KMT2ACYP2C9CYP2C19
SCHEMBL8567515 0.81 VCP (0.41) ALDH1A1CYP2C9CYP2C19SMN1; SMN2CYP1A2
Hydrochloric Acid SCHEMBL8563542 0.78 ALDH1A1 (0.39) ALDH1A1MEN1KMT2ACYP2C9CYP2C19
SCHEMBL8560120 0.71 ALDH1A1 (0.38) ALDH1A1KMT2ACYP2C9CYP2C19SMN1; SMN2
SCHEMBL9051616 0.69 ALDH1A1 (0.40) ALDH1A1CYP2C9CYP2C19TSHRL3MBTL1
SCHEMBL7015162 0.69 ALDH1A1 (0.58) ALDH1A1MEN1KMT2ACYP2C9CYP2C19
SCHEMBL8562859 0.67 ALDH1A1 (0.38) ALDH1A1CYP2C9CYP2C19SMN1; SMN2CYP1A2
SCHEMBL7219920 0.64 ALDH1A1 (0.52) ALDH1A1MEN1KMT2ACYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0552060-B1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO (JP) 1998-11-18 EP disclosed
EP-0700911-A1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO., LTD. (JP) 1996-03-13 EP disclosed
US-5472965-A Useful for treatment of retrovirus infections; less toxic SHIONOGI & CO., LTD. (JP) 1995-12-05 US disclosed
US-5326780-A Acquired immunodeficiency syndrome SHIONOGI & CO., LTD. (JP) 1994-07-05 US disclosed
EP-0552060-A1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO., LTD. (JP) 1993-07-21 EP disclosed