SCHEMBL8568157

SCHEMBL8568157

CCc1noc2cccc(N3CCN(Cc4ccccc4)CC3)c12

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 8/20 0.49
DRD2 P14416 7/20 0.49
DRD3 P35462 6/20 0.49
ACHE P22303 3/20 0.46
HTR1A P08908 1/20 0.46
MAPT P10636 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
NCF1 P14598 1/20 0.44
SIGMAR1 Q99720 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8574032 0.79 ACHE (0.52) ACHE
SCHEMBL12000243 0.73 DRD4 (0.64) DRD4DRD2DRD3MAPTNPSR1
Maleic Acid SCHEMBL8574182 0.73 ACHE (0.49) DRD2ACHESIGMAR1
Fumaric Acid SCHEMBL8574186 0.73 ACHE (0.49) DRD2ACHESIGMAR1
SCHEMBL8569904 0.70 ACHE (0.53) ACHE
SCHEMBL13533025 0.69 HTR1A (0.83) DRD2HTR1A
SCHEMBL8131885 0.69 ATM (0.67) DRD4DRD2DRD3NCF1SIGMAR1
SCHEMBL6986033 0.69 ACHE (0.70) ACHESIGMAR1
SCHEMBL6864941 0.68 DRD4 (0.81) DRD4DRD2DRD3SIGMAR1
Hydrochloric Acid SCHEMBL6991446 0.68 ACHE (0.68) ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750542-A Benzisoxazole and benzisothizole derivatives as cholinesterase inhibitors PFIZER (US) 1998-05-12 US disclosed