SCHEMBL8570497

SCHEMBL8570497

CNC(=O)C(C)Oc1cc(-c2nn(C)c(C(F)(F)F)c2Cl)c(F)cc1Cl

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 5/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 2/20 0.34
SMN1; SMN2 Q16637 4/20 0.34
RORC P51449 1/20 0.34
MAPT P10636 2/20 0.33
HPGD P15428 2/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
MEN1 O00255 1/20 0.33
ALOX12 P18054 1/20 0.33
TP53 P04637 1/20 0.33
ERBB2 P04626 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6911659 0.89 PTGDR2 (0.37) ALDH1A1KDM4ETSHRRORCHPGD
SCHEMBL9696140 0.84 LMNA (0.34) GAAALDH1A1KDM4ELMNATSHR
SCHEMBL6912537 0.83 MEN1 (0.33) KMT2AMEN1
SCHEMBL27304825 0.83 PPOX (0.37)
SCHEMBL6909705 0.80 BACE1 (0.35) GAAALDH1A1KDM4ELMNAMAPK1
SCHEMBL5398257 0.78 CYP1A2 (0.35) KMT2AMAPTMEN1
SCHEMBL27321856 0.78 MAPT (0.31) KMT2ASMN1; SMN2MAPTMEN1
SCHEMBL6909703 0.77 PKM (0.44) ALDH1A1KDM4ETSHRRORCHPGD
SCHEMBL27320851 0.75 MAPT (0.34) GAAALDH1A1LMNASMN1; SMN2MAPT
SCHEMBL9857297 0.75 PPOX (0.36) GAAALDH1A1KDM4ELMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1050121-C Process for preparing substituted aryl-halogenoalkyl pyrazoles MONSANTO CO (US) 2000-03-08 CN disclosed
EP-0553307-B1 HERBICIDAL SUBSTITUTED ARYL-HALOALKYLPYRAZOLES MONSANTO CO (US) 1998-12-09 EP disclosed
EP-0791571-A1 Benzoyl derivatives MONSANTO COMPANY (US) 1997-08-27 EP disclosed
US-5536700-A Herbicidal compositions comprising aryl-5-haloalkylpyrazoles and glyphosate, it's salts, diquat or paraquat MONSANTO COMPANY (US) 1996-07-16 US disclosed
US-5530126-A ALKYLATION IN INERT SOLVENT MONSANTO COMPANY (US) 1996-06-25 US disclosed
US-5496956-A BY ESTERIFICATION OF CARBOXY SUBSTITUTION WITH ALCOHOLS IN THE PRESENCE OF MINERAL ACID MONSANTO COMPANY (US) 1996-03-05 US disclosed
US-5489571-A CROP-SAFE COMPOUNDS EFFECTIVE AT LOW CONCENTRATIONS MONSANTO COMPANY (US) 1996-02-06 US disclosed
CN-1030595-C Substituted aryl-haloalkyl-pyrazoles as herbicides MONSANTO CO (US) 1996-01-03 CN disclosed
US-5281571-A Herbicidal benzoxazinone- and benzothiazinone-substituted pyrazoles MONSANTO COMPANY (US) 1994-01-25 US disclosed
EP-0553307-A1 HERBICIDAL SUBSTITUTED ARYL-HALOALKYLPYRAZOLES MONSANTO COMPANY (US) 1993-08-04 EP disclosed
WO-1992006962-A1 HERBICIDAL SUBSTITUTED ARYL-HALOALKYLPYRAZOLES MONSANTO COMPANY (US) 1992-04-30 WO disclosed