SCHEMBL8575158

SCHEMBL8575158

COc1cc(OC)c(C(=O)CCCCCl)cc1Cl

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 8/20 0.51
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
HTR2B P41595 1/20 0.46
ALDH1A1 P00352 2/20 0.44
ACHE P22303 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8574455 0.89 KMT2A (0.50) HTR4HTR2AHTR2CHTR2B
SCHEMBL7357981 0.87 HTR4 (0.67) HTR4ALDH1A1ACHEGAA
SCHEMBL8569585 0.84 HTR4 (0.50) HTR4ALDH1A1ACHEGAA
SCHEMBL7355259 0.83 AGER (0.53) HTR4ALDH1A1SMN1; SMN2LMNAHPGD
SCHEMBL11836438 0.81 STING1 (0.57) HTR4ALDH1A1ACHE
SCHEMBL6702779 0.81 MEN1 (0.52) HTR4HTR2AHTR2CHTR2BALDH1A1
SCHEMBL8571105 0.81 HTR2A (0.55) HTR2AHTR2CHTR2BALDH1A1LMNA
SCHEMBL8572360 0.81 HTR2A (0.54) HTR4HTR2AHTR2CHTR2BALDH1A1
SCHEMBL17844481 0.80 STING1 (0.46) HTR4ALDH1A1ACHESMN1; SMN2LMNA
SCHEMBL8572525 0.79 ALDH1A1 (0.56) ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739336-A SELECTIVE 5-HYDROXYTRYPTAMINE-2C RECEPTOR ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1998-04-14 US disclosed
WO-1997000872-A1 1,3,8-TRIAZA- AND 3,8-DIAZA-1-OXASPIRO(4,5)DECANE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 1997-01-09 WO disclosed