SCHEMBL8569585

SCHEMBL8569585

COc1cc(OC)c(C(=O)CCCCCl)cc1N

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 9/20 0.50
GAA P10253 2/20 0.41
ACHE P22303 2/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40
KMT2A Q03164 1/20 0.40
CYP3A4 P08684 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC1 Q13547 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8574455 0.88 KMT2A (0.50) HTR4MEN1KMT2ACYP3A4HDAC8
SCHEMBL7357981 0.86 HTR4 (0.67) HTR4GAAACHEMEN1ALDH1A1
SCHEMBL8575158 0.84 HTR4 (0.51) HTR4GAAACHEALDH1A1
SCHEMBL8572525 0.78 ALDH1A1 (0.56) MEN1ALDH1A1KMT2AHDAC8HDAC1
SCHEMBL8570776 0.78 ALDH1A1 (0.42) HTR4MEN1ALDH1A1KMT2ACYP3A4
SCHEMBL8571284 0.77 RAB9A (0.58) MEN1ALDH1A1KMT2AHDAC1
SCHEMBL8571105 0.77 HTR2A (0.55) MEN1ALDH1A1TSHRKMT2A
SCHEMBL8572360 0.77 HTR2A (0.54) HTR4MEN1ALDH1A1KMT2AHDAC8
SCHEMBL8569807 0.77 KMT2A (0.53) MEN1ALDH1A1TSHRKMT2AHDAC8
SCHEMBL29156702 0.76 KDM4E (0.50) HTR4GAAACHEALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739336-A SELECTIVE 5-HYDROXYTRYPTAMINE-2C RECEPTOR ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1998-04-14 US disclosed
WO-1997000872-A1 1,3,8-TRIAZA- AND 3,8-DIAZA-1-OXASPIRO(4,5)DECANE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 1997-01-09 WO disclosed