SCHEMBL8576753

SCHEMBL8576753

COc1ccc(Cn2c(=O)[nH]c(=O)c3[nH]c(C4CCCC4)nc32)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 4/20 0.60
ADORA2A P29274 4/20 0.59
ADORA2B P29275 4/20 0.59
ADORA3 P0DMS8 3/20 0.53
HPGD P15428 4/20 0.49
ALDH1A1 P00352 4/20 0.49
KDM4E B2RXH2 2/20 0.49
TLR7 Q9NYK1 2/20 0.49
GAA P10253 1/20 0.49
MAPT P10636 1/20 0.49
HTT P42858 1/20 0.49
KMT2A Q03164 3/20 0.48
NPSR1 Q6W5P4 1/20 0.48
PNP P00491 1/20 0.47
MEN1 O00255 2/20 0.45
GMNN O75496 1/20 0.45
LMNA P02545 1/20 0.45
CYP1A2 P05177 1/20 0.45
TSHR P16473 1/20 0.45
PMP22 Q01453 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8579120 0.90 ADORA1 (0.64) ADORA1ADORA2AADORA2BADORA3HPGD
SCHEMBL8579881 0.88 ADORA1 (0.62) ADORA1ADORA2AADORA2BADORA3HPGD
SCHEMBL8355232 0.87 ADORA3 (0.65) ADORA1ADORA2AADORA2BADORA3HPGD
SCHEMBL6094064 0.78 KMT2A (0.70) ADORA3HPGDALDH1A1KDM4ETLR7
SCHEMBL8580800 0.78 ADORA1 (0.76) ADORA1ADORA2AADORA2BADORA3KMT2A
SCHEMBL8575318 0.77 ADORA1 (0.65) ADORA1ADORA2AADORA2BADORA3KMT2A
SCHEMBL8118476 0.76 ADORA1 (1.00) ADORA1ADORA2AADORA2BADORA3KMT2A
SCHEMBL8578121 0.76 ADORA1 (0.72) ADORA1ADORA2AADORA2BADORA3KMT2A
SCHEMBL8020381 0.75 ADORA2B (0.68) ADORA1ADORA2AADORA2BADORA3KMT2A
SCHEMBL8579784 0.75 ADORA1 (0.65) ADORA1ADORA2AADORA2BADORA3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1043348-C Asymmetrically substituted xanthines BOEHRINGER INGELHEIM KG (DE) 1999-05-12 CN disclosed
US-5719279-A CHOLINOMIMETICS BOEHRINGER INGELHEIM KG (DE) 1998-02-17 US disclosed
EP-0654033-A1 ASYMMETRICALLY SUBSTITUTED XANTHINE WITH ADENOSINE-ANTAGONISTIC PROPERTIES BOEHRINGER INGELHEIM KG (DE) 1995-05-24 EP disclosed
WO-1994003456-A1 ASYMMETRICALLY SUBSTITUTED XANTHINE WITH ADENOSINE-ANTAGONISTIC PROPERTIES BOEHRINGER INGELHEIM KG (DE) 1994-02-17 WO disclosed