SCHEMBL8583345

SCHEMBL8583345

COC(=O)c1ccc(C2CCCC2C)c(S(C)(=O)=O)c1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.36
HSD17B10 Q99714 5/20 0.36
TSHR P16473 4/20 0.36
HPGD P15428 2/20 0.36
KDM4E B2RXH2 8/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
TAS1R2 Q8TE23 1/20 0.34
NPSR1 Q6W5P4 2/20 0.34
KMT2A Q03164 2/20 0.33
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33
DRD3 P35462 1/20 0.33
HTR5A P47898 1/20 0.33
LMNA P02545 2/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA5A P35218 1/20 0.33
CA9 Q16790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8583100 0.87 FFAR4 (0.38) ALDH1A1HSD17B10HPGDKDM4ESMN1; SMN2
SCHEMBL8578771 0.86 TAS1R3 (0.37) ALDH1A1HSD17B10TSHRHPGDKDM4E
SCHEMBL8583191 0.86 KDM4E (0.36) ALDH1A1HSD17B10TSHRHPGDKDM4E
SCHEMBL8582996 0.84 KDM4E (0.37) ALDH1A1HSD17B10TSHRHPGDKDM4E
SCHEMBL27367149 0.83 TAS1R3 (0.32) TAS1R3TAS1R1TAS1R2LMNAHTT
SCHEMBL8581355 0.83 ALDH1A1 (0.36) ALDH1A1KDM4ESMN1; SMN2KMT2AYAP1
SCHEMBL8581200 0.83 ALOX5AP (0.37) ALDH1A1HSD17B10TSHRHPGDKDM4E
SCHEMBL8579296 0.82 PDK2 (0.39) ALDH1A1HSD17B10TSHRHPGDKDM4E
SCHEMBL8578782 0.82 DRD2 (0.38) ALDH1A1HSD17B10TSHRHPGDKDM4E
SCHEMBL8580134 0.81 YAP1 (0.39) ALDH1A1HSD17B10TSHRHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5840761-A Alkylbenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-11-24 US disclosed