SCHEMBL8586983

SCHEMBL8586983

COc1ccccc1C1(O)CC2CCC(C1)N2C

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 4/20 0.61
SLC6A3 Q01959 4/20 0.61
SLC6A2 P23975 3/20 0.61
ALDH1A1 P00352 1/20 0.58
TSHR P16473 1/20 0.58
DRD2 P14416 1/20 0.56
DRD3 P35462 1/20 0.56
HTR1A P08908 3/20 0.53
SIGMAR1 Q99720 1/20 0.51
OPRM1 P35372 3/20 0.50
OPRL1 P41146 3/20 0.50
OPRD1 P41143 2/20 0.50
OPRK1 P41145 2/20 0.50
CHRM2 P08172 1/20 0.49
CHRM4 P08173 1/20 0.49
CHRM5 P08912 1/20 0.49
CHRM1 P11229 1/20 0.49
CHRM3 P20309 1/20 0.49
SLC6A1 P30531 1/20 0.43
SLC6A12 P48065 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10008740 0.81 DRD2 (0.64) SLC6A4SLC6A3SLC6A2ALDH1A1TSHR
SCHEMBL1267331 0.79 ALDH1A1 (0.55) SLC6A4SLC6A3SLC6A2ALDH1A1TSHR
SCHEMBL6747981 0.77 SIGMAR1 (0.56) ALDH1A1TSHRDRD2DRD3HTR1A
SCHEMBL31028212 0.74 OPRM1 (0.46) SLC6A4SLC6A3SLC6A2ALDH1A1TSHR
SCHEMBL5194656 0.74 SLC6A4 (0.74) SLC6A4SLC6A3SLC6A2ALDH1A1DRD2
SCHEMBL5193526 0.72 ALDH1A1 (0.52) SLC6A4SLC6A3SLC6A2ALDH1A1DRD2
SCHEMBL29965651 0.72 SIGMAR1 (0.72) ALDH1A1TSHRDRD2DRD3SIGMAR1
SCHEMBL7542807 0.72 SIGMAR1 (0.72) ALDH1A1TSHRDRD2DRD3SIGMAR1
SCHEMBL5566258 0.71 SLC6A4 (0.64) SLC6A4SLC6A3SLC6A2ALDH1A1OPRM1
SCHEMBL5349498 0.70 SIGMAR1 (0.70) ALDH1A1TSHRSIGMAR1OPRM1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0819126-A1 BIPHENYLAMIDE DERIVATIVES AS 5HT 1D? ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1998-01-21 EP disclosed
WO-1996031508-A1 BIPHENYLAMIDE DERIVATIVES AS 5HT1D ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1996-10-10 WO disclosed