SCHEMBL8587138

SCHEMBL8587138

CC(C)Oc1ccc(-c2ccnc(N3CCC(CN)C3)n2)cc1C(C)(C)C

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DKK1 O94907 3/20 0.52
RBP4 P02753 6/20 0.39
KMO O15229 2/20 0.37
SYK P43405 1/20 0.36
ROCK2 O75116 3/20 0.36
ROCK1 Q13464 2/20 0.36
TTR P02766 3/20 0.36
AAK1 Q2M2I8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8511678 0.94 DKK1 (0.58) DKK1RBP4KMOROCK2ROCK1
SCHEMBL8514887 0.93 DKK1 (0.45) DKK1KMOAAK1
SCHEMBL8515838 0.88 DKK1 (0.49) DKK1KMOROCK2
Ammonia Solution, Strong SCHEMBL8587136 0.86 DYRK1A (0.43) DKK1RBP4KMO
SCHEMBL8512439 0.86 DKK1 (0.56) DKK1KMOROCK2
Hydrochloric Acid SCHEMBL8513412 0.85 DKK1 (0.55) DKK1KMOROCK2
SCHEMBL8510671 0.85 DKK1 (0.44) DKK1KMO
SCHEMBL8514134 0.82 DKK1 (0.42) DKK1KMO
SCHEMBL8510840 0.81 KMO (0.43) DKK1KMO
SCHEMBL8510734 0.81 ZAP70 (0.41) DKK1KMOROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed