SCHEMBL8587459

SCHEMBL8587459

CCCNS(=O)(=O)C(C)(C)c1ccc(-c2ccsc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRIA4 P48058 2/20 0.44
IDH2 P48735 2/20 0.37
GRIA2 P42262 3/20 0.36
KCNH2 Q12809 1/20 0.35
CNR1 P21554 1/20 0.35
CYP2E1 P05181 1/20 0.34
CYP2A6 P11509 1/20 0.34
CYP2B6 P20813 1/20 0.34
NPY5R Q15761 2/20 0.34
MAP3K5 Q99683 1/20 0.34
CYP17A1 P05093 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
CYP1A2 P05177 1/20 0.33
GSK3B P49841 1/20 0.33
FYN P06241 1/20 0.33
DRD3 P35462 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8587550 0.89 GRIA4 (0.46) GRIA4IDH2GRIA2KCNH2CNR1
SCHEMBL8585627 0.83 NPY5R (0.37) IDH2NPY5RCYP11B1CYP11B2FYN
SCHEMBL8585587 0.82 IDH2 (0.37) GRIA4IDH2GRIA2NPY5RFYN
SCHEMBL8583844 0.82 KIF11 (0.46)
SCHEMBL8585276 0.81 ALDH1A1 (0.40) GRIA4
SCHEMBL7570581 0.81 CA12 (0.43) GRIA4DRD3
SCHEMBL8586293 0.80 CA12 (0.51) GRIA4CNR1CYP1A2
SCHEMBL8585567 0.80 L3MBTL1 (0.43)
SCHEMBL8587469 0.80 KIF11 (0.51)
SCHEMBL8585612 0.80

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998033496-A1 SULPHONAMIDE DERIVATIVES ELI LILLY AND COMPANY (US) 1998-08-06 WO disclosed