SCHEMBL8587702

SCHEMBL8587702

CC(C)(C)[C@H](N)C(=O)N(C(=O)OCc1ccccc1)[C@H](C=O)Cc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSB P07858 3/20 0.42
ABCB1 P08183 2/20 0.39
ALDH1A1 P00352 1/20 0.38
SLC15A1 P46059 2/20 0.37
LTA4H P09960 2/20 0.37
LAP3 P28838 1/20 0.37
CTSL P07711 1/20 0.36
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
SLC1A3 P43003 2/20 0.36
SLC1A2 P43004 2/20 0.36
SLC1A1 P43005 2/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1151902 0.87 CTSB (0.46) CTSBABCB1ALDH1A1SLC15A1LTA4H
SCHEMBL8586153 0.87 CTSB (0.45) CTSBABCB1ALDH1A1SLC15A1LTA4H
SCHEMBL8586501 0.87 CTSB (0.39) CTSBABCB1ALDH1A1SLC15A1LTA4H
SCHEMBL8583695 0.86 SLC15A1 (0.45) CTSBABCB1ALDH1A1SLC15A1LTA4H
SCHEMBL8583463 0.84 EPHX1 (0.40) CTSBABCB1ALDH1A1SLC15A1LTA4H
SCHEMBL8586822 0.84 CTSB (0.43) CTSBABCB1SLC15A1LTA4HLAP3
SCHEMBL8586811 0.83 CTSB (0.47) CTSBABCB1SLC15A1LTA4HCTSL
SCHEMBL8584621 0.82 CTSB (0.41) CTSBABCB1SLC15A1CTSLCTSS
SCHEMBL8583834 0.82 SLC15A1 (0.40) CTSBABCB1SLC15A1LTA4HLAP3
SCHEMBL9714126 0.80 ALOX5 (0.42) CTSBALDH1A1SLC15A1CTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0840614-A1 CALPAIN INHIBITORS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES SANOFI WINTHROP, INC. (US) 1998-05-13 EP claimed
WO-1996041638-A1 CALPAIN INHIBITORS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES SANOFI WINTHROP, INC. (US) 1996-12-27 WO claimed