SCHEMBL8587732

SCHEMBL8587732

COc1cc2scc(CCN)c2cc1OC

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 6/20 0.46
KDM4E B2RXH2 1/20 0.46
ATM Q13315 1/20 0.46
HTR2A P28223 6/20 0.44
HTR2C P28335 2/20 0.44
ADRA1A P35348 1/20 0.44
HTR2B P41595 1/20 0.43
CYP1A2 P05177 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9123944 0.88 TAAR1 (0.58) TAAR1KDM4EATMHTR2AHTR2C
SCHEMBL3480270 0.81 MAOA (0.47) TAAR1
SCHEMBL10663751 0.81 POLB (0.49) ATMHTR2A
SCHEMBL8587828 0.78 TAAR1 (0.53) TAAR1HTR2AHTR2CADRA1ACYP1A2
SCHEMBL8586269 0.78 MTNR1A (0.61) TAAR1HTR2AHTR2CADRA1ACYP1A2
SCHEMBL5547193 0.73 MAOA (0.41) KDM4E
SCHEMBL5547192 0.73 MAOA (0.41)
SCHEMBL9751556 0.71 CA2 (0.56) TAAR1HTR2ACYP1A2
SCHEMBL8586513 0.71 TAAR1 (0.53) TAAR1KDM4EATMHTR2AADRA1A
SCHEMBL73404 0.71 TAAR1 (0.53) TAAR1HTR2AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998027984-A1 METHOD OF PRODUCING ANALGESIA BY ADMINISTRATION OF 1,2,3,4-TETRAHYDROBENZO-[b]THIENO[2,3-c]PYRIDINE AND DERIVATIVES NEUREX CORPORATION (US) 1998-07-02 WO disclosed
US-4971974-A ANOREXIGENIC AGENTS, BENZO B!THIENO 2,3-C!PYRIDINE COMPOUNDS NEUREX CORPORATION (US) 1990-11-20 US disclosed