SCHEMBL8587828

SCHEMBL8587828

COc1ccc2c(CCN)csc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.53
ADRA1A P35348 1/20 0.53
HTR2A P28223 2/20 0.52
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
HTR1D P28221 2/20 0.49
HTR6 P50406 2/20 0.49
MAPT P10636 2/20 0.49
CYP1A2 P05177 2/20 0.49
HTR1A P08908 1/20 0.49
TSHR P16473 1/20 0.49
NFKB1 P19838 1/20 0.49
HTR1B P28222 1/20 0.49
HTR2C P28335 1/20 0.49
HTR7 P34969 1/20 0.49
HTR4 Q13639 1/20 0.49
TRPM8 Q7Z2W7 1/20 0.49
MTNR1A P48039 5/20 0.48
MTNR1B P49286 4/20 0.48
BLM P54132 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8586269 0.88 MTNR1A (0.61) TAAR1ADRA1AHTR2AMEN1KMT2A
SCHEMBL5541597 0.86 MTNR1A (0.49) HTR2AKMT2AMAPTTSHRMTNR1A
SCHEMBL10663900 0.82 MTNR1A (0.55) HTR2AHTR6MAPTMTNR1AMTNR1B
SCHEMBL10470119 0.82 MTNR1A (0.52) HTR2AMEN1KMT2AMAPTMTNR1A
SCHEMBL6839987 0.81 CYP2A6 (0.53) MAPTTSHRMTNR1AMTNR1BNPSR1
SCHEMBL5439262 0.81 MTNR1A (0.44) MAPTTSHRMTNR1AMTNR1BNPSR1
SCHEMBL5544113 0.81 MTNR1A (0.51) HTR2AMEN1KMT2AMAPTMTNR1A
SCHEMBL5211436 0.81 PPARG (0.46) MEN1KMT2AHTR1AMTNR1AMTNR1B
SCHEMBL8021641 0.79 MTNR1A (0.59) TAAR1ADRA1AHTR2AMEN1KMT2A
SCHEMBL10663910 0.79 HTR2A (0.55) TAAR1HTR2AHTR1AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998027984-A1 METHOD OF PRODUCING ANALGESIA BY ADMINISTRATION OF 1,2,3,4-TETRAHYDROBENZO-[b]THIENO[2,3-c]PYRIDINE AND DERIVATIVES NEUREX CORPORATION (US) 1998-07-02 WO disclosed
US-4971974-A ANOREXIGENIC AGENTS, BENZO B!THIENO 2,3-C!PYRIDINE COMPOUNDS NEUREX CORPORATION (US) 1990-11-20 US disclosed
US-4764506-A IMMUNOINFLAMMATION WARNER-LAMBERT COMPANY (US) 1988-08-16 US disclosed
US-4636493-A HYPOTENSIVES WARNER-LAMBERT COMPANY (US) 1987-01-13 US disclosed
US-4600707-A ANTIPSYCHOTIC AGENTS, HYPOTENSIVES WARNER-LAMBERT COMPANY (US) 1986-07-15 US disclosed