SCHEMBL8588488

SCHEMBL8588488

[C]1C=NOc2ccccc2C1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31
OXTR P30559 1/20 0.31
ABCG2 Q9UNQ0 1/20 0.30
ITGB2 P05107 1/20 0.30
ICAM1 P05362 1/20 0.30
ITGAL P20701 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5550 0.71 MAOA (0.38) MAOAMAOBGAAOXTRABCG2
SCHEMBL31513481 0.68 MAOA (0.39) MAOAMAOBLMNAGAAOXTR
SCHEMBL8925 0.68 MAOA (0.39) MAOAMAOBLMNAGAAOXTR
SCHEMBL3928581 0.68 MAOA (0.39) MAOAMAOBLMNAGAAOXTR
SCHEMBL7679301 0.67 MAOA (0.38) MAOAMAOBGAAOXTRABCG2
Hydrochloric Acid SCHEMBL8707066 0.67 MAOA (0.38) MAOAMAOBGAAOXTRABCG2
Hydrochloric Acid SCHEMBL8699855 0.67 MAOA (0.38) MAOAMAOBGAAOXTRABCG2
Water SCHEMBL15284972 0.67 MAOA (0.38) MAOAMAOBGAAOXTRABCG2
Methylamine SCHEMBL6415772 0.64 MAOA (0.35) MAOAMAOBKDM4ENPC1ALDH1A1
SCHEMBL3074959 0.64 MAOA (0.50) MAOAMAOBKDM4ENPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2643317-A1 BENZOXAZEPINES AS INHIBITORS OF P13K/MTOR AND METHODS OF THEIR USE AND MANUFACTURE Exelixis, Inc. (US) 2013-10-02 EP disclosed
WO-2012071519-A1 BENZOXAZEPINES AS INHIBITORS OF P13K/MTOR AND METHODS OF THEIR USE AND MANUFACTURE EXELIXIS, INC. (US) 2012-05-31 WO disclosed