SCHEMBL3928581

SCHEMBL3928581

[C]1[CH]Oc2ccccc2C1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOA P21397 7/20 0.39
MAOB P27338 7/20 0.39
ABCG2 Q9UNQ0 1/20 0.33
ITGB2 P05107 1/20 0.33
ICAM1 P05362 1/20 0.33
ITGAL P20701 1/20 0.33
OXTR P30559 1/20 0.33
IDO1 P14902 2/20 0.32
GAA P10253 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
AOC2 O75106 5/20 0.31
DAO P14920 1/20 0.31
LMNA P02545 2/20 0.30
CRHBP P24387 2/20 0.30
CRHR2 Q13324 2/20 0.30
SMN1; SMN2 Q16637 2/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL105430 0.73 MAOA (0.39) MAOAMAOBABCG2ITGB2ICAM1
SCHEMBL8588488 0.68 MAOA (0.35) MAOAMAOBABCG2ITGB2ICAM1
SCHEMBL3128 0.67
SCHEMBL2851479 0.67
SCHEMBL5550 0.67 MAOA (0.38) MAOAMAOBABCG2ITGB2ICAM1
SCHEMBL5065 0.64 MAOA (0.39) MAOAMAOBABCG2ITGB2ICAM1
SCHEMBL453819 0.64 MAOA (0.39) MAOAMAOBABCG2ITGB2ICAM1
SCHEMBL241643 0.64 OXTR (0.42) MAOAMAOBABCG2ITGB2ICAM1
SCHEMBL450202 0.64 MAOA (0.39) MAOAMAOBABCG2ITGB2ICAM1
SCHEMBL1289715 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7557130-B2 Bicyclic heteroaromatic alanines UCB PHARMA, S.A. (BE) 2009-07-07 US disclosed
US-20040209913-A1 e.g., 3-[1-(3,5-Dichloroisonicotinoyl)-2,3-dihydro-1 H-indol-5-yl]-2-[(3-oxo-spiro[3.5]non-1-en-1-yl)amino]-propanoate; modulating cell adhesion for the prophylaxis or treatment of inflammatory diseases or disorders, such as rheumatoid arthritis, in which the extravasculation of leukocytes plays a role. UCB PHARMA S.A. (BE) 2004-10-21 US disclosed
WO-2003011815-A1 BICYCLIC HETEROAROMATIC ALANINES CELLTECH R & D LIMITED (GB) 2003-02-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040209913-A1 e.g., 3-[1-(3,5-Dichloroisonicotinoyl)-2,3-dihydro-1 H-indol-5-yl]-2-[(3-oxo-spiro[3.5]non-1-en-1-yl)amino]-propanoate; modulating cell adhesion for the prophylaxis or treatment of inflammatory diseases or disorders, such as rheumatoid arthritis, in which the extravasculation of leukocytes plays a role. ICAM1, VCAM1, CCR1 MAOA 2507/4885MAOB 2742/4885ABCG2 1991/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.