SCHEMBL8596052

SCHEMBL8596052

COc1ccc(C#N)c(-c2ccccc2)c1OC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 2/20 0.53
IMPDH1 P20839 1/20 0.53
MAOA P21397 1/20 0.51
MAOB P27338 1/20 0.51
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 1/20 0.45
USP2 O75604 1/20 0.45
AR P10275 6/20 0.43
PGR P06401 2/20 0.43
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
ADORA2A P29274 2/20 0.42
ADORA1 P30542 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
USP8 P40818 1/20 0.40
USP7 Q93009 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7575609 0.80 IMPDH2 (0.53) IMPDH2IMPDH1MAOAMAOBALDH1A1
SCHEMBL16109256 0.80 PDE4B (0.53) ALDH1A1KDM4EUSP2PDE4APDE4B
SCHEMBL28684149 0.79 AR (0.50) IMPDH2IMPDH1MAOAMAOBAR
SCHEMBL6988623 0.78 PDE4A (0.42) MAOAMAOBPDE4APDE4BPDE4C
SCHEMBL27608025 0.78 IMPDH2 (0.47) IMPDH2IMPDH1ALDH1A1KDM4EUSP2
SCHEMBL7274689 0.76 SMN1; SMN2 (0.42) MAOAMAOBALDH1A1KDM4EPDE4A
SCHEMBL3432260 0.76 IMPDH2 (0.49) IMPDH2IMPDH1MAOAMAOBALDH1A1
SCHEMBL4696500 0.76 ALDH1A1 (0.55) IMPDH2IMPDH1MAOAMAOBALDH1A1
SCHEMBL29123961 0.76 MAOB (0.57) IMPDH2IMPDH1MAOAMAOBALDH1A1
SCHEMBL3643547 0.75 NPC1 (0.54) ALDH1A1KDM4EUSP2PDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0877734-A1 QUINOLINE AND QUINAZOLINE COMPOUNDS USEFUL IN THERAPY Pfizer Research and Development Company, N.V./S.A. (IE) 1998-11-18 EP disclosed
WO-1997023462-A1 QUINOLINE AND QUINAZOLINE COMPOUNDS USEFUL IN THERAPY PFIZER RESEARCH AND DEVELOPMENT COMPANY, N.V./S.A. (IE) 1997-07-03 WO disclosed