SCHEMBL7274689

SCHEMBL7274689

COc1ccc(CC#N)c(-c2ccccc2)c1OC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
POLB P06746 2/20 0.41
PDE4A P27815 2/20 0.40
PDE4B Q07343 2/20 0.40
PDE4C Q08493 2/20 0.40
PDE4D Q08499 2/20 0.40
KDM4E B2RXH2 4/20 0.38
HPGD P15428 3/20 0.38
MAPT P10636 3/20 0.38
GAA P10253 1/20 0.38
ALDH1A1 P00352 4/20 0.38
HTT P42858 1/20 0.37
IDO1 P14902 1/20 0.37
TDO2 P48775 1/20 0.37
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7279625 0.87 ALDH1A1 (0.41) SMN1; SMN2NPC1RAB9APOLBKDM4E
SCHEMBL7281786 0.80 PDE4B (0.47) SMN1; SMN2NPC1RAB9APOLBPDE4A
SCHEMBL6234576 0.79 AOC3 (0.49) SMN1; SMN2POLBKDM4EMAPTGAA
SCHEMBL7274265 0.78 PDE4B (0.39) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL7274263 0.77 POLB (0.46) SMN1; SMN2POLBKDM4EHPGDGAA
SCHEMBL7282980 0.77 SMN1; SMN2 (0.40) SMN1; SMN2NPC1RAB9APOLBKDM4E
SCHEMBL8596052 0.76 IMPDH2 (0.53) SMN1; SMN2NPC1RAB9APOLBPDE4A
SCHEMBL16109256 0.76 PDE4B (0.53) SMN1; SMN2NPC1RAB9APOLBPDE4A
Hydrochloric Acid SCHEMBL7272763 0.76 TAAR1 (0.51)
SCHEMBL9786028 0.76 AOC3 (0.39) SMN1; SMN2POLBKDM4EMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4885313-A 3,4-Dihydroxyphenylethylamine derivatives and their use FISONS PLC (GB) 1989-12-05 US disclosed
US-4803225-A Dihydroxy-phenethylamino compounds useful as pharmaceuticals FISONS, PLC (GB) 1989-02-07 US disclosed
US-4720586-A Substituted 3,4-dihydroxy-phenylethylamino compounds FISONS, PLC (GB) 1988-01-19 US disclosed
EP-0142283-A2 Phenylethylamines, process for their preparation and compositions containing them FISONS plc (GB) 1985-05-22 EP disclosed