SCHEMBL8596702

SCHEMBL8596702

NNC(=O)Nc1ccc2ccccc2c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.71
NPC1 O15118 5/20 0.71
MAPT P10636 3/20 0.71
CA2 P00918 2/20 0.62
CA12 O43570 1/20 0.59
CA1 P00915 1/20 0.59
CA9 Q16790 1/20 0.59
MEN1 O00255 5/20 0.59
KMT2A Q03164 5/20 0.59
POLB P06746 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.59
CYP1A2 P05177 2/20 0.56
ALDH1A1 P00352 2/20 0.56
KDM4E B2RXH2 1/20 0.56
CYP2C19 P33261 1/20 0.56
HIF1A Q16665 1/20 0.56
EPHX1 P07099 3/20 0.54
LMNA P02545 1/20 0.54
TDP1 Q9NUW8 1/20 0.53
GAA P10253 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9547503 0.88 RAB9A (0.89) RAB9ANPC1MAPTCA2CA12
SCHEMBL30697002 0.83 MAPT (1.00) RAB9ANPC1MAPTCA2CA12
SCHEMBL11049543 0.83 MAPT (1.00) RAB9ANPC1MAPTCA2CA12
SCHEMBL8325083 0.81 RAB9A (0.71) RAB9ANPC1MAPTCA2CA12
SCHEMBL516845 0.81 RAB9A (0.65) RAB9ANPC1MAPTCA2CA12
SCHEMBL24272501 0.80 MAPT (0.80) RAB9ANPC1MAPTCA2CA12
SCHEMBL24272500 0.80 MAPT (0.80) RAB9ANPC1MAPTCA2CA12
SCHEMBL14470404 0.79 NPC1 (0.77) RAB9ANPC1MAPTCA2CA12
SCHEMBL11057371 0.79 NPC1 (0.77) RAB9ANPC1MAPTCA2CA12
SCHEMBL1672113 0.79 RAB9A (0.72) RAB9ANPC1MAPTCA2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726314-A ACETYLCHOLINESTERASE INHIBITORS AS NERVE AGENT ANTIDOTES GEORGIA TECH RESEARCH CORP. (US) 1998-03-10 US disclosed
US-5714615-A ACETYLCHOLINESTERASE ENZYME INHIBITOR, STIMULATE NICOTINIC RECEPTORS IN CENTRAL NERVOUS SYSTEM GEORGIA TECH RESEARCH CORPORATION (US) 1998-02-03 US disclosed
WO-1995021822-A1 PYRIDINIUM COMPOUNDS GEORGIA TECH RESEARCH CORPORATION (US) 1995-08-17 WO disclosed
US-5290942-A Acetylcholinesterase inhibitors GEORGIA TECH RESEARCH CORPORATION (US) 1994-03-01 US disclosed
US-5206371-A Acetylcholinesterase inhibitor GEORGIA TECH RESEARCH CORPORATION (US) 1993-04-27 US disclosed
US-5180831-A Acetylcholinesterase Inhibitors GEORGIA TECH RESEARCH CORPORATION (US) 1993-01-19 US disclosed