SCHEMBL8599412

SCHEMBL8599412

Cc1ccc2c(c1)C(=O)CC21CCCCC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.54
ATM Q13315 3/20 0.54
HTT P42858 1/20 0.54
RAD52 P43351 1/20 0.38
PGR P06401 1/20 0.37
METAP1 P53582 2/20 0.37
ACHE P22303 1/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
PARP1 P09874 1/20 0.36
PARP10 Q53GL7 1/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
KMT2A Q03164 1/20 0.35
ELANE P08246 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8601620 0.98 KDM4E (0.53) KDM4EATMHTTRAD52PGR
SCHEMBL13001156 0.81 KDM4E (0.40) KDM4EATMHTTHRH3ALDH1A1
SCHEMBL27212869 0.80 KDM4E (0.43) KDM4EATMHTTRAD52PGR
SCHEMBL29341252 0.80 S100A4 (0.37) KDM4EATMHTTMETAP1CA1
SCHEMBL11545783 0.78 HDAC4 (0.37) ACHECA1CA2CA7CA9
SCHEMBL11547924 0.78 PDE7A (0.42) PGRMETAP1PARP1PARP10ALDH1A1
SCHEMBL29341181 0.78 S100A4 (0.38) KDM4EMETAP1CA1CA2CA4
SCHEMBL11542025 0.78 MEN1 (0.38) KDM4EATMHTTCA9PARP1
SCHEMBL11544646 0.78 PBRM1 (0.44) KDM4ECA1CA2CA7CA9
SCHEMBL8596234 0.78 GRIN1 (0.46) KDM4EMETAP1ACHECA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0657426-B1 Tricyclic pyrrole derivatives HOFFMANN LA ROCHE (CH) 1998-07-22 EP disclosed
US-5646173-A ANTISEROTONINE AGENTS; CENTRAL NERVOUS SYSTEM DISORDERS; ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1997-07-08 US disclosed