SCHEMBL8596234

SCHEMBL8596234

COc1ccc2c(c1)C(=O)CC21CCCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.46
GRIN2A Q12879 1/20 0.46
GRIN2B Q13224 1/20 0.46
PDE7A Q13946 2/20 0.46
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
KDM4E B2RXH2 3/20 0.43
KLK7 P49862 1/20 0.43
METAP1 P53582 2/20 0.42
ACHE P22303 1/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
ALDH1A1 P00352 4/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
PRNP P04156 1/20 0.39
PPIB P23284 1/20 0.39
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31649958 0.83 GRIN1 (0.45) GRIN1GRIN2AGRIN2BPDE7APDE3B
SCHEMBL11819676 0.80 PDE3B (0.47) PDE7APDE3BPDE3AKDM4EKLK7
SCHEMBL31650373 0.79 ACHE (0.46) GRIN1GRIN2AGRIN2BPDE7APDE3B
SCHEMBL8597253 0.79 PDE3B (0.47) PDE3BPDE3AKDM4EKLK7METAP1
SCHEMBL8601620 0.79 KDM4E (0.53) KDM4EMETAP1ACHECA1CA2
SCHEMBL8599412 0.78 KDM4E (0.54) KDM4EMETAP1ACHECA1CA2
SCHEMBL11547924 0.76 PDE7A (0.42) PDE7AMETAP1ALDH1A1
SCHEMBL11544646 0.76 PBRM1 (0.44) KDM4ECA1CA2CA7CA9
SCHEMBL11545783 0.76 HDAC4 (0.37) ACHECA1CA2CA7CA9
SCHEMBL29341181 0.76 S100A4 (0.38) KDM4EMETAP1CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0657426-B1 Tricyclic pyrrole derivatives HOFFMANN LA ROCHE (CH) 1998-07-22 EP disclosed
US-5646173-A ANTISEROTONINE AGENTS; CENTRAL NERVOUS SYSTEM DISORDERS; ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1997-07-08 US disclosed
US-4172093-A Pharmacodynamically active indan derivatives AB KABI (SE) 1979-10-23 US disclosed