SCHEMBL8599469

SCHEMBL8599469

COc1ccc(-c2cc(-c3cccc(CN)n3)nc(-c3cccc(CNCC(=O)O)n3)c2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
LTB4R Q15722 3/20 0.42
MCL1 Q07820 2/20 0.40
ADORA3 P0DMS8 2/20 0.40
PTGS2 P35354 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
SCN9A Q15858 1/20 0.38
GYS1 P13807 1/20 0.38
EGLN1 Q9GZT9 1/20 0.37
ERCC5 P28715 1/20 0.37
FEN1 P39748 1/20 0.37
MAPK1 P28482 1/20 0.36
FYN P06241 1/20 0.36
CASP3 P42574 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8935842 0.95 ALDH1A1 (0.47) ALDH1A1KDM4EHPGDSMN1; SMN2LTB4R
SCHEMBL8633585 0.87 HPGD (0.41) ALDH1A1KDM4EHPGDSMN1; SMN2LTB4R
SCHEMBL7847605 0.84 ABL1 (0.44) SMN1; SMN2MCL1ADORA3MAPK1CASP3
SCHEMBL8596932 0.82 MCL1 (0.41) ALDH1A1KDM4EHPGDSMN1; SMN2LTB4R
SCHEMBL7771784 0.77 HSP90AA1 (0.45) KDM4ESMN1; SMN2ADORA2AADORA1LMNA
SCHEMBL8765283 0.76 MCL1 (0.45) ALDH1A1KDM4EHPGDSMN1; SMN2LTB4R
SCHEMBL8596986 0.75 ABL1 (0.44) ALDH1A1KDM4ESMN1; SMN2LTB4RMCL1
SCHEMBL13217240 0.74 MCL1 (0.42) ALDH1A1KDM4EHPGDSMN1; SMN2LTB4R
Acetic Acid SCHEMBL27847203 0.74 MCL1 (0.40) SMN1; SMN2MCL1LMNAHTTSCN9A
SCHEMBL8935757 0.74 ADORA3 (0.43) ALDH1A1KDM4EHPGDSMN1; SMN2LTB4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5744119-A LABELING A PROTEIN/TERPYRIDINE COMPLEX WITH A METAL RADIONUCLIDE STERLING WINTHROP (US) 1998-04-28 US disclosed
US-5539117-A 2-acetyl-6-cyanopyridines and their use as intermediates in the synthesis of oligo-2,6-pyridines GE HEALTHCARE AS (NO) 1996-07-23 US disclosed