SCHEMBL8633585

SCHEMBL8633585

COc1ccc(-c2cc(-c3cccc(CNCC(=O)O)n3)nc(-c3cccc(CN(CC(=O)O)CC(=O)O)n3)c2)cc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
LTB4R Q15722 3/20 0.41
AVPR1B P47901 2/20 0.39
MCL1 Q07820 2/20 0.39
ADORA3 P0DMS8 2/20 0.38
PTGER2 P43116 3/20 0.38
PTGS2 P35354 1/20 0.36
GYS1 P13807 1/20 0.36
MEP1A Q16819 1/20 0.36
MEP1B Q16820 1/20 0.36
EGLN1 Q9GZT9 1/20 0.36
ERCC5 P28715 1/20 0.35
FEN1 P39748 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8935842 0.92 ALDH1A1 (0.47) HPGDKDM4EALDH1A1SMN1; SMN2LTB4R
SCHEMBL8765283 0.91 MCL1 (0.45) HPGDKDM4EALDH1A1SMN1; SMN2LTB4R
SCHEMBL13217240 0.88 MCL1 (0.42) HPGDKDM4EALDH1A1SMN1; SMN2LTB4R
SCHEMBL8599469 0.87 ALDH1A1 (0.43) HPGDKDM4EALDH1A1SMN1; SMN2LTB4R
SCHEMBL8596932 0.86 MCL1 (0.41) HPGDKDM4EALDH1A1SMN1; SMN2LTB4R
SCHEMBL8597039 0.84 MEN1 (0.44) KDM4ELTB4RMCL1ADORA3PTGER2
SCHEMBL8935826 0.81 ADORA3 (0.46) KDM4EALDH1A1LTB4RAVPR1BADORA3
SCHEMBL13997749 0.80 LTB4R (0.39) KDM4EALDH1A1LTB4RMCL1ADORA3
SCHEMBL8935762 0.79 KMT2A (0.43) HPGDKDM4EALDH1A1SMN1; SMN2MCL1
SCHEMBL8601997 0.79 ALDH1A1 (0.44) HPGDKDM4EALDH1A1SMN1; SMN2ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5744119-A LABELING A PROTEIN/TERPYRIDINE COMPLEX WITH A METAL RADIONUCLIDE STERLING WINTHROP (US) 1998-04-28 US disclosed
US-5539117-A 2-acetyl-6-cyanopyridines and their use as intermediates in the synthesis of oligo-2,6-pyridines GE HEALTHCARE AS (NO) 1996-07-23 US disclosed
US-5350696-A 2-acetyl-6-cyanopyridines and their use as intermediates in the synthesis of oligo-2,6-pyridines STERLING WINTHROP, INC. (US) 1994-09-27 US disclosed