SCHEMBL8599840

SCHEMBL8599840

CCCCN1C(=O)COc2cc(F)c(N)cc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 3/20 0.51
CHRM5 P08912 2/20 0.51
CHRM3 P20309 2/20 0.51
REN P00797 1/20 0.40
EGFR P00533 4/20 0.39
SLC5A1 P13866 1/20 0.39
SLC5A2 P31639 1/20 0.39
POLB P06746 1/20 0.39
SCN9A Q15858 1/20 0.39
GAA P10253 1/20 0.38
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38
CYP1A2 P05177 1/20 0.38
HTR1A P08908 1/20 0.38
CYP2C9 P11712 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8598261 0.96 CHRM1 (0.50) CHRM1CHRM5CHRM3RENEGFR
SCHEMBL8602365 0.92 CHRM1 (0.47) CHRM1CHRM5CHRM3RENEGFR
SCHEMBL29901598 0.88 CHRM1 (0.46) CHRM1CHRM5CHRM3RENEGFR
SCHEMBL8600207 0.87 RORC (0.43) CHRM1CHRM5CHRM3POLB
SCHEMBL10592910 0.85 CHRM1 (0.45) CHRM1CHRM5CHRM3RENEGFR
SCHEMBL29901589 0.85 CHRM1 (0.43) CHRM1CHRM5CHRM3EGFR
SCHEMBL29901581 0.84 REN (0.44) CHRM1CHRM5CHRM3RENDRD2
SCHEMBL8878855 0.81 CHRM1 (0.41) CHRM1CHRM5CHRM3SLC5A1SLC5A2
SCHEMBL10431134 0.80 HTT (0.47) CHRM1POLBCYP1A2CYP2C19
SCHEMBL8600208 0.79 CYP11B2 (0.42) CHRM1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626370-B1 Process for producing aromatic isothiocyanate derivatives SUMITOMO CHEMICAL CO (JP) 1998-02-11 EP disclosed
EP-0626370-A1 Process for producing aromatic isothiocyanate derivatives SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1994-11-30 EP disclosed