SCHEMBL8601016

SCHEMBL8601016

CN(C(=O)Cl)c1cccc(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.49
HSD17B1 P14061 1/20 0.48
HSD17B2 P37059 1/20 0.48
RXFP1 Q9HBX9 2/20 0.47
CES2 O00748 1/20 0.47
ALDH1A1 P00352 1/20 0.47
TACR1 P25103 2/20 0.46
MAPT P10636 3/20 0.45
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
POLQ O75417 1/20 0.45
POLB P06746 1/20 0.43
RXRA P19793 1/20 0.43
RXRB P28702 1/20 0.43
RXRG P48443 1/20 0.43
P2RX1 P51575 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28141847 0.85 TP53 (0.50) TP53HSD17B1HSD17B2RXFP1CES2
SCHEMBL11174926 0.85 TACR1 (0.50) TP53HSD17B1HSD17B2RXFP1CES2
SCHEMBL10943479 0.83 TP53 (0.49) TP53HSD17B1HSD17B2RXFP1CES2
SCHEMBL14955365 0.83 POLQ (0.51) TP53HSD17B1HSD17B2RXFP1CES2
SCHEMBL1118844 0.82 PTGIR (0.46) TP53CES2TACR1MAPTHTT
SCHEMBL9835938 0.81 CES2 (0.49) TP53CES2ALDH1A1MAPTHTT
SCHEMBL9835457 0.81 CES2 (0.49) TP53CES2ALDH1A1MAPTHTT
SCHEMBL7675880 0.81 TP53 (0.54) TP53HSD17B1HSD17B2RXFP1CES2
SCHEMBL12220665 0.81 RXFP1 (0.54) TP53HSD17B1HSD17B2RXFP1CES2
SCHEMBL11402034 0.81 POLQ (0.52) TP53HSD17B1HSD17B2RXFP1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5767286-A REACTING A TETRAZOLINONE WITH A CARBAMOYL CHLORIDE IN THE PRESENCE OF 4-DIMETHYLAMINOPYRIDINE NIHON BAYER AGROCHEM K. K. (JP) 1998-06-16 US disclosed
EP-0646577-B1 Process for the preparation of 1,4-disubstituted-5(4H)-tetrazolinones BAYER AGROCHEM KK (JP) 1998-06-03 EP disclosed
EP-0646577-A1 Process for the preparation of 1,4-disubstituted-5(4H)-tetrazolinones NIHON BAYER AGROCHEM K.K. (JP) 1995-04-05 EP disclosed
US-4046909-A Pyrrolidylidene, piperidylidene and hexahydroazepinylidene ureas as CNS depressants MCNEIL LABORATORIES, INCORPORATED (US) 1977-09-06 US disclosed
US-3998958-A Pyrrolidylidene, piperidylidene and hexahydroazepinylidene ureas as CNS depressants MCNEIL LABORATORIES, INCORPORATED (US) 1976-12-21 US disclosed