SCHEMBL8601137

SCHEMBL8601137

O=[N+](O)c1ccc(COP([O-])(O)=S)cc1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.53
IDO1 P14902 2/20 0.39
PGK1 P00558 1/20 0.37
PGK2 P07205 1/20 0.37
TSHR P16473 3/20 0.37
MAOB P27338 1/20 0.36
ALDH1A1 P00352 2/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
PLA2G4B P0C869 1/20 0.33
RAB9A P51151 2/20 0.33
HTR2A P28223 1/20 0.33
NPC1 O15118 1/20 0.33
CYP3A4 P08684 1/20 0.33
MAPK1 P28482 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5983777 0.85 AKR1C3 (0.58) AKR1C3IDO1PGK1PGK2TSHR
SCHEMBL5331963 0.78 AKR1C3 (0.67) AKR1C3IDO1PGK1PGK2TSHR
SCHEMBL1024521 0.74 CA1 (0.49) AKR1C3TSHRALDH1A1CA1CA2
SCHEMBL11378806 0.73 AKR1C3 (0.46) AKR1C3IDO1PGK1PGK2TSHR
SCHEMBL735220 0.72 AKR1C3 (0.44) AKR1C3IDO1PGK1PGK2TSHR
SCHEMBL2374254 0.72 AKR1C3 (0.42) AKR1C3IDO1PGK1PGK2TSHR
SCHEMBL3625606 0.69 TSHR (0.42) AKR1C3TSHRALDH1A1RAB9ANPC1
SCHEMBL5983772 0.69 AKR1C3 (0.81) AKR1C3IDO1PGK1PGK2TSHR
SCHEMBL6209548 0.69 CA2 (0.42) AKR1C3IDO1TSHRMAOBALDH1A1
SCHEMBL5069158 0.69 AKR1C3 (1.00) AKR1C3IDO1PGK1PGK2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0723973-B1 Nucleoside phosphorothioate derivatives, synthesis and use thereof KING S COLLEGE LONDON (GB) 1998-10-21 EP disclosed
US-5708161-A Nucleoside phosphorothioate derivatives, synthesis and use thereof KING'S COLLEGE LONDON (GB) 1998-01-13 US disclosed
EP-0723973-A1 Nucleoside phosphorothioate derivatives, synthesis and use thereof KING'S COLLEGE LONDON (GB) 1996-07-31 EP disclosed