SCHEMBL8604402

SCHEMBL8604402

COc1ccc(-c2nc(CNC(=O)NO)oc2-c2ccccc2S(N)(=O)=O)cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.43
PTGS1 P23219 4/20 0.43
RXRA P19793 3/20 0.40
SCN9A Q15858 2/20 0.39
EPHX2 P34913 1/20 0.37
NR4A2 P43354 3/20 0.37
AURKA O14965 1/20 0.37
ROCK2 O75116 1/20 0.37
RPS6KA5 O75582 1/20 0.37
NTRK1 P04629 1/20 0.37
LCK P06239 1/20 0.37
CSF1R P07333 1/20 0.37
LYN P07948 1/20 0.37
RET P07949 1/20 0.37
KIT P10721 1/20 0.37
FGFR1 P11362 1/20 0.37
FER P16591 1/20 0.37
FLT1 P17948 1/20 0.37
RPS6KB1 P23443 1/20 0.37
FLT4 P35916 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6315580 0.89 PTGS2 (0.45) PTGS2PTGS1RXRASCN9AEPHX2
SCHEMBL8604021 0.87 PTGS1 (0.41) PTGS2PTGS1RXRAEPHX2NR4A2
SCHEMBL8604398 0.86 PTGS2 (0.48) PTGS2PTGS1RXRAEPHX2RXRB
SCHEMBL6308151 0.85 PTGS2 (0.48) PTGS2PTGS1RXRAEPHX2NR4A2
SCHEMBL8604310 0.85 RXRA (0.43) RXRANR4A2RXRBRXRGF10
SCHEMBL6309069 0.83 NR4A2 (0.49) PTGS2PTGS1RXRAEPHX2NR4A2
SCHEMBL7520783 0.83 AURKA (0.45) PTGS2PTGS1AURKAROCK2RPS6KA5
SCHEMBL8561125 0.83 PTGS2 (0.47) PTGS2PTGS1RXRASCN9AEPHX2
SCHEMBL6307441 0.82 PTGS2 (0.44) PTGS2PTGS1RXRAEPHX2NR4A2
SCHEMBL6309656 0.82 NR4A2 (0.51) PTGS2PTGS1RXRAEPHX2NR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828718-A1 HETEROCYCLO SUBSTITUTED HYDROXAMIC ACID DERIVATIVES AS CYCLOOXYGENASE-2 AND 5-LIPOXYGENASE INHIBITORS G.D. SEARLE & CO. (US) 1998-03-18 EP disclosed
WO-1996038418-A1 HETEROCYCLO SUBSTITUTED HYDROXAMIC ACID DERIVATIVES AS CYCLOOXYGENASE-2 AND 5-LIPOXYGENASE INHIBITORS G.D. SEARLE & CO. (US) 1996-12-05 WO disclosed