SCHEMBL8604398

SCHEMBL8604398

COc1ccc(-c2nc(CNC(=O)NO)oc2-c2ccc(S(N)(=O)=O)cc2)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.48
PTGS1 P23219 11/20 0.48
ALDH1A1 P00352 2/20 0.40
EPHX2 P34913 1/20 0.39
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39
NLRP3 Q96P20 1/20 0.38
NAMPT P43490 1/20 0.38
LMNA P02545 1/20 0.38
PPARD Q03181 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8605996 0.91 PTGS2 (0.47) PTGS2PTGS1ALDH1A1EPHX2RXRA
SCHEMBL6315576 0.88 PTGS2 (0.50) PTGS2PTGS1ALDH1A1EPHX2RXRA
SCHEMBL8604016 0.86 CA2 (0.44) PTGS2PTGS1EPHX2RXRARXRB
SCHEMBL8604402 0.86 PTGS2 (0.43) PTGS2PTGS1EPHX2RXRARXRB
SCHEMBL6308148 0.84 PTGS2 (0.51) PTGS2PTGS1EPHX2RXRARXRB
SCHEMBL8604308 0.84 RXRA (0.47) PTGS2PTGS1ALDH1A1RXRARXRB
SCHEMBL8605984 0.84 RXRA (0.47) PTGS2PTGS1ALDH1A1RXRARXRB
SCHEMBL6309066 0.82 PTGS2 (0.49) PTGS2PTGS1EPHX2RXRARXRB
SCHEMBL8606213 0.82 PTGS2 (0.53) PTGS2PTGS1ALDH1A1NLRP3LMNA
SCHEMBL7520779 0.81 PTGS2 (0.47) PTGS2PTGS1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828718-A1 HETEROCYCLO SUBSTITUTED HYDROXAMIC ACID DERIVATIVES AS CYCLOOXYGENASE-2 AND 5-LIPOXYGENASE INHIBITORS G.D. SEARLE & CO. (US) 1998-03-18 EP disclosed
WO-1996038418-A1 HETEROCYCLO SUBSTITUTED HYDROXAMIC ACID DERIVATIVES AS CYCLOOXYGENASE-2 AND 5-LIPOXYGENASE INHIBITORS G.D. SEARLE & CO. (US) 1996-12-05 WO disclosed