SCHEMBL8604772

SCHEMBL8604772

NS(=O)(=O)c1ccc(-c2csc(CNC(=O)NO)c2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.44
PTGS1 P23219 1/20 0.44
CA1 P00915 7/20 0.43
CA2 P00918 7/20 0.43
CA12 O43570 6/20 0.43
CA9 Q16790 5/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
ALDH1A1 P00352 1/20 0.42
ALOX12 P18054 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
KDM4E B2RXH2 2/20 0.42
GAA P10253 1/20 0.42
HTT P42858 1/20 0.42
CHRNA7 P36544 2/20 0.41
IKBKB O14920 2/20 0.40
CHUK O15111 2/20 0.40
CA7 P43166 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8604775 0.84 F10 (0.38) PTGS2PTGS1CA2CA9
SCHEMBL8606779 0.78 KDM4E (0.44) PTGS2PTGS1CA1CA2CA12
SCHEMBL6316750 0.77 PTGS1 (0.45) PTGS2PTGS1CA1CA2CA12
SCHEMBL6050650 0.75 PTGS2 (0.56) PTGS2PTGS1CA1CA2CA12
SCHEMBL6314458 0.74 PTGS2 (0.42) PTGS2PTGS1CA1CA2CA12
SCHEMBL6314888 0.74 CHRNA7 (0.41) PTGS2PTGS1CA1CA2CA12
SCHEMBL6309619 0.70 PTGS2 (0.50) PTGS2PTGS1CA2
SCHEMBL7070547 0.69 PTGS2 (0.70) PTGS2PTGS1CA1CA2CA9
SCHEMBL6315334 0.69 CA1 (0.39) PTGS2PTGS1CA1CA2CA12
SCHEMBL8604308 0.69 RXRA (0.47) PTGS2PTGS1CA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828718-A1 HETEROCYCLO SUBSTITUTED HYDROXAMIC ACID DERIVATIVES AS CYCLOOXYGENASE-2 AND 5-LIPOXYGENASE INHIBITORS G.D. SEARLE & CO. (US) 1998-03-18 EP disclosed
WO-1996038418-A1 HETEROCYCLO SUBSTITUTED HYDROXAMIC ACID DERIVATIVES AS CYCLOOXYGENASE-2 AND 5-LIPOXYGENASE INHIBITORS G.D. SEARLE & CO. (US) 1996-12-05 WO disclosed