SCHEMBL8604308

SCHEMBL8604308

NS(=O)(=O)c1ccc(-c2oc(CNC(=O)NO)nc2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 3/20 0.47
RXRB P28702 3/20 0.47
RXRG P48443 3/20 0.47
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
PTGS1 P23219 4/20 0.43
PTGS2 P35354 4/20 0.43
CA2 P00918 8/20 0.43
CA1 P00915 7/20 0.43
CA9 Q16790 7/20 0.43
CA12 O43570 6/20 0.43
CA4 P22748 2/20 0.42
CA7 P43166 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NR4A2 P43354 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ALOX12 P18054 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8605984 1.00 RXRA (0.47) RXRARXRBRXRGMAOAMAOB
SCHEMBL8606984 0.90 RXRA (0.50) RXRARXRBRXRGMAOAMAOB
SCHEMBL8607283 0.89 PTGS2 (0.57) MAOAMAOBPTGS1PTGS2CA2
SCHEMBL8606384 0.89 RXRA (0.47) RXRARXRBRXRGPTGS1PTGS2
SCHEMBL8604016 0.88 CA2 (0.44) RXRARXRBRXRGMAOAMAOB
SCHEMBL6308845 0.86 RXRA (0.49) RXRARXRBRXRGMAOAMAOB
SCHEMBL6310934 0.86 RXRA (0.49) RXRARXRBRXRGMAOAMAOB
SCHEMBL8604398 0.84 PTGS2 (0.48) RXRARXRBRXRGPTGS1PTGS2
SCHEMBL8605986 0.84 RXRA (0.43) RXRARXRBRXRGCA2CA9
SCHEMBL8604310 0.84 RXRA (0.43) RXRARXRBRXRGCA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828718-A1 HETEROCYCLO SUBSTITUTED HYDROXAMIC ACID DERIVATIVES AS CYCLOOXYGENASE-2 AND 5-LIPOXYGENASE INHIBITORS G.D. SEARLE & CO. (US) 1998-03-18 EP disclosed
WO-1996038418-A1 HETEROCYCLO SUBSTITUTED HYDROXAMIC ACID DERIVATIVES AS CYCLOOXYGENASE-2 AND 5-LIPOXYGENASE INHIBITORS G.D. SEARLE & CO. (US) 1996-12-05 WO disclosed