SCHEMBL8605151

SCHEMBL8605151

CC(C)(C)OC(=O)N(CC(=O)O)Cc1ccccc1N

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
NCOR2 Q9Y618 1/20 0.40
CTSL P07711 2/20 0.38
CTSB P07858 2/20 0.38
CTSS P25774 2/20 0.38
KDM4E B2RXH2 1/20 0.36
AKT1 P31749 2/20 0.36
KEAP1 Q14145 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP2C19 P33261 1/20 0.35
HIF1A Q16665 1/20 0.35
FDPS P14324 1/20 0.34
SSTR4 P31391 1/20 0.34
RECQL P46063 1/20 0.33
BACE1 P56817 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3406057 0.86 HDAC3 (0.39) HDAC3HDAC1HDAC2NCOR2CTSL
SCHEMBL21257785 0.84 ALDH1A1 (0.38) HDAC3HDAC1HDAC2NCOR2KDM4E
SCHEMBL18322690 0.84 ALDH1A1 (0.40) HDAC3HDAC1HDAC2NCOR2CTSL
SCHEMBL3402058 0.83 SLC6A4 (0.37) HDAC3HDAC1HDAC2NCOR2KEAP1
SCHEMBL2834319 0.82 HDAC3 (0.55) HDAC3HDAC1HDAC2NCOR2CTSL
SCHEMBL21257736 0.82 HDAC3 (0.35) HDAC3HDAC1HDAC2NCOR2CTSL
SCHEMBL12330698 0.81 ALDH1A1 (0.42)
SCHEMBL27829838 0.81 HDAC3 (0.37) HDAC3HDAC1HDAC2NCOR2CTSL
SCHEMBL7211228 0.80 FDPS (0.37) HDAC3HDAC1HDAC2NCOR2KDM4E
SCHEMBL2061803 0.80 SLC6A4 (0.43) HDAC3HDAC1HDAC2NCOR2CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108112251-B NRF2 modulators 葛兰素史克知识产权发展有限公司 2021-03-05 CN disclosed
EP-0789571-A4 CYCLIC AMIDINE ANALOGS AS INHIBITORS OF NITRIC OXIDE SYNTHASE MERCK & CO INC (US) 1999-04-14 EP disclosed
EP-0789571-A1 CYCLIC AMIDINE ANALOGS AS INHIBITORS OF NITRIC OXIDE SYNTHASE Merck & Co., Inc. (US) 1997-08-20 EP disclosed