SCHEMBL8606563

SCHEMBL8606563

CSc1cc(Cl)ccc1C(=CC#N)OC(=O)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX1 P51575 4/20 0.35
P2RX4 Q99571 2/20 0.35
P2RX7 Q99572 2/20 0.35
TMPRSS4 Q9NRS4 2/20 0.35
GABRA1 P14867 2/20 0.35
GABRG2 P18507 2/20 0.35
GABRB3 P28472 2/20 0.35
GABRB1 P18505 1/20 0.35
GABRB2 P47870 1/20 0.35
DDR1 Q08345 2/20 0.33
MEN1 O00255 1/20 0.33
IKBKB O14920 1/20 0.33
CHUK O15111 1/20 0.33
KDR P35968 1/20 0.33
FLT3 P36888 1/20 0.33
KMT2A Q03164 1/20 0.33
MYLK Q15746 1/20 0.33
MAP4K5 Q9Y4K4 1/20 0.33
CLPP Q16740 1/20 0.33
RHOC P08134 5/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9412822 0.74 P2RX1 (0.38) P2RX1P2RX4P2RX7TMPRSS4DDR1
SCHEMBL8607647 0.72 P2RX1 (0.38) P2RX1P2RX4P2RX7TMPRSS4DDR1
SCHEMBL14893085 0.64 CES2 (0.64) P2RX1RHOCRHOANOTUM
SCHEMBL8608917 0.62 KMT2A (0.49) GABRA1GABRG2GABRB3GABRB1GABRB2
SCHEMBL10334495 0.62 SMN1; SMN2 (0.57) MEN1KMT2ANOTUM
SCHEMBL8607500 0.62 SMN1; SMN2 (0.42) MEN1KDRKMT2A
SCHEMBL5274963 0.62 CES2 (0.55) P2RX1MEN1KMT2ANOTUM
SCHEMBL8017606 0.62 MAOB (0.42) MEN1KDRKMT2A
SCHEMBL5843160 0.61 CFTR (0.63) MEN1KMT2ANOTUM
SCHEMBL4096751 0.60 KDM4E (0.50) GABRA1GABRG2GABRB3GABRB2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5804532-A REACTING A BENZOYL ISOXAZOLE WITH A BASE RHONE-POULENC AGRICULTURE LIMITED (GB) 1998-09-08 US disclosed
EP-0625505-A2 2-Cyano-1,3-dione derivatives and their use as herbicides RHONE POULENC AGRICULTURE LTD. (GB) 1994-11-23 EP disclosed