SCHEMBL8608561

SCHEMBL8608561

CSc1cc(C(=O)C(C#N)C(=O)C2CC2)ccc1C

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 4/20 0.39
TAS1R1 Q7RTX1 4/20 0.39
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
SLC6A3 Q01959 2/20 0.32
HRH3 Q9Y5N1 2/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31
MEN1 O00255 1/20 0.31
CYP2D6 P10635 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8608718 0.79 SMN1; SMN2 (0.39) RAB9AKMT2A
SCHEMBL8609169 0.78 MGLL (0.30) KDM4EALDH1A1MAPTRAB9A
SCHEMBL8607183 0.75
SCHEMBL8607103 0.74 CTSK (0.35) KDM4EALDH1A1RAB9AMEN1CYP2D6
SCHEMBL14155670 0.74 NPC1 (0.38) TAS1R3TAS1R1KDM4ERAB9AMEN1
SCHEMBL8953567 0.73 GSK3B (0.51) SLC6A3KDM4EALDH1A1RAB9A
SCHEMBL9237726 0.72 ALDH1A1 (0.48) ALDH1A1MAPTRAB9AMEN1CYP2D6
SCHEMBL9119216 0.72 PRKCI (0.45) TAS1R3TAS1R1RAB9A
SCHEMBL8048258 0.71
SCHEMBL1224446 0.71 MGLL (0.41) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0625508-B1 Sulfur-containing derivatives of 2-cyano-1,3-diones and their use as herbicides RHONE POULENC AGRICULTURE (GB) 1998-08-19 EP claimed
EP-0625508-A2 Sulfur-containing derivatives of 2-cyano-1,3-diones and their use as herbicides RHONE POULENC AGRICULTURE LTD. (GB) 1994-11-23 EP claimed
JP-6329620-A None JP disclosed
US-5804532-A REACTING A BENZOYL ISOXAZOLE WITH A BASE RHONE-POULENC AGRICULTURE LIMITED (GB) 1998-09-08 US disclosed
EP-0625508-B1 Sulfur-containing derivatives of 2-cyano-1,3-diones and their use as herbicides RHONE POULENC AGRICULTURE (GB) 1998-08-19 EP disclosed
JP-H06329620-A NOVEL HERBICIDE RHONE POULENC AGRICULTURE LTD 1994-11-29 JP disclosed
EP-0625508-A2 Sulfur-containing derivatives of 2-cyano-1,3-diones and their use as herbicides RHONE POULENC AGRICULTURE LTD. (GB) 1994-11-23 EP disclosed