SCHEMBL8610216

SCHEMBL8610216

COC(=O)c1cc(OC(F)(F)F)ccc1F.NC(N)=NC(=O)c1cc(OC(F)(F)F)ccc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.39
ABL1 P00519 2/20 0.38
CFTR P13569 1/20 0.37
SLC9A1 P19634 2/20 0.37
BRAF P15056 1/20 0.36
PDK2 Q15119 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.36
SCN9A Q15858 1/20 0.36
CHEK1 O14757 1/20 0.36
FFAR1 O14842 1/20 0.36
FFAR4 Q5NUL3 1/20 0.36
EPHX2 P34913 1/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
LCLAT1 Q6UWP7 1/20 0.35
PIM1 P11309 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9018732 0.92 FFAR4 (0.40) ABL1SLC9A1BRAFKMT2ACHEK1
SCHEMBL8611570 0.88 CFTR (0.40) MRGPRX4ABL1CFTRALDH1A1KMT2A
SCHEMBL17478821 0.87 ABL1 (0.45) MRGPRX4ABL1CFTRBRAFALDH1A1
SCHEMBL8610122 0.85 SLC9A1 (0.40) MRGPRX4CFTRSLC9A1
SCHEMBL8611439 0.84 CFTR (0.53) MRGPRX4CFTRSLC9A1PDK2KDM4E
SCHEMBL8614188 0.83 MRGPRX4 (0.40) MRGPRX4CFTRSLC9A1KMT2AKDM4E
SCHEMBL8614095 0.83 MRGPRX4 (0.38) MRGPRX4ABL1CFTRSLC9A1CHEK1
SCHEMBL8612520 0.82 SLC9A1 (0.40) MRGPRX4SLC9A1
SCHEMBL9018666 0.81 PIM1 (0.40) SLC9A1KMT2ACHEK1FFAR1FFAR4
SCHEMBL9018694 0.80 SLC9A1 (0.44) SLC9A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5747539-A Fluorine-containing benzoylguanidines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-05-05 US disclosed